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[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-3-yl]methanol
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yloxy)acetamide
1-(3-chlorophenyl)-4-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]piperazin-2-one
2-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpiperidine-3-carboxamide
N-(1-hydroxy-2-methylpropan-2-yl)-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[2-(pyrazin-2-yl)ethyl]piperidine-3-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-benzofuran-7-carboxamide
(1S,6R)-9-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3,9-diazabicyclo[4.2.1]nonane
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-6-ethoxy-1,2-dihydroquinolin-2-one
3-(5-{2-[(2-methylphenyl)sulfanyl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(3-methylpyridin-2-yl)methyl]piperidin-4-ol
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(thiophen-3-ylmethyl)piperazine
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(furan-3-ylmethyl)piperidine
(3S,4R)-4-phenyl-1-{[(1s,4s)-4-aminocyclohexyl]methyl}pyrrolidine-3-carboxylic acid
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidine
N-(1-methyl-1H-pyrazol-5-yl)-2-[3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
(5S)-5-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
3-(1-{[5-(methylcarbamoyl)furan-2-yl]methyl}piperidin-3-yl)benzoic acid
2-(4-ethoxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
2-amino-6-(propan-2-yl)-N-[3-(pyridin-4-yl)propyl]pyrimidine-4-carboxamide
5-chloro-N-(2-methoxyethyl)-N-methyl-3-phenyl-1H-indole-2-carboxamide
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
2-(azepan-1-yl)-N-(2-methanesulfonamidoethyl)acetamide
2-{1-[(1-ethylpyrrolidin-2-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-1,3-benzodiazole
2-(2-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
1-(1'-{[4-(methylsulfanyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
{[7-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl}(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-(2-chlorophenyl)-N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]furan-2-carboxamide
1-(2,2-difluorocyclopropanecarbonyl)-4-phenoxypiperidine-4-carboxylic acid
7-(5-chloropyridin-2-yl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(4-{[1-(hydroxymethyl)-9-propyl-3,9-diazaspiro[5.5]undecan-3-yl]methyl}thiophen-2-yl)ethan-1-one
3-(3-methoxyphenoxymethyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
methyl 3-(cyclobutylmethoxy)-5-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]benzoate
2-{[3-(cyclopropylmethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]methyl}-2H-1,2,3-benzotriazole
N-(3-methyl-1H-pyrazol-5-yl)-2-(9-methyl-9H-carbazol-3-yl)acetamide
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-hexyl-8-(3-hydroxypyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-2-(pyridin-3-yl)acetamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)cyclopropanesulfonamide
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyrimidin-2-amine
6-({8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(3-chlorophenyl)ethyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}acetamide
8-methoxy-2-(thiophen-3-yl)quinoline