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3-methyl-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-1-propyl-1H-pyrazole-4-carboxamide
N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-(3-methoxyphenyl)azetidine-1-carboxamide
2-[(3-methoxyphenyl)sulfanyl]-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]ethan-1-one
4-(3-ethylphenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2,5-dimethoxyphenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
4-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-3-yl)benzoic acid
2-(4-chloro-2-methoxybenzoyl)-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
2-{[(3,5-dimethylphenyl)methyl]sulfanyl}-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
1-[2-(1H-pyrazol-1-yl)benzoyl]-4-(pyridin-3-ylmethyl)piperazine
3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
(2E)-1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(pent-4-enoyl)piperidine-3-carboxylate
(2S,4S)-4-amino-N-ethyl-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
5-methyl-7-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}pyrazolo[1,5-a]pyrimidine
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
2-(2,5-dimethoxyphenyl)-5-methyl-4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}-1,3-oxazole
(2S,4R)-4-amino-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
6-(dimethylamino)-N-[2-(3-phenylpiperidin-1-yl)ethyl]pyridine-3-carboxamide
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
2,2-dimethyl-5-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]thiomorpholin-3-one
7-[(4-fluorophenyl)methyl]-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(2R,3S,6R)-5-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(3-fluoro-4-methoxyphenyl)-N-[(4-fluorophenyl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-{4-azaspiro[2.5]octan-4-ylmethyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
2-({methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}methyl)benzonitrile
6-methyl-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-6-methoxyphenol
2-{[3-(morpholin-4-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
2-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}quinolin-4-ol
2-[4-(dimethylamino)phenyl]-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
methyl 2-(azocane-1-sulfonyl)-6-(3-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-(4-aminopyrimidin-2-yl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-(2-phenoxyacetyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-[(3S,4R)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
dimethyl[(5-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}thiophen-3-yl)methyl]amine
2-ethyl-N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-6-methylpyrimidin-4-amine
1-{4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}ethan-1-one
2-{1-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
N'-cyclopentyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}butanediamide
3-[(3R,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-butyl-3-hydroxy-4-methoxy-N-(3-phenylprop-2-yn-1-yl)benzamide
{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
1-(4-fluoro-3-methylbenzoyl)-2-(3-methoxypropyl)piperidine
1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-(dimethylamino)-2-(2-fluorophenyl)-N-(oxan-4-yl)acetamide
1-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-2-[(4-methoxyphenyl)methyl]-1H-1,3-benzodiazole