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2-(2-chloro-6-methoxyphenyl)-5-propylpyrimidine
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[(3-fluoro-4-methylphenyl)methyl]amine
1-(cyclopropylmethyl)-5-[(3-methylthiophen-2-yl)sulfonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-methoxy-2-{[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}phenol
3-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
[(2-cyclohexylpyrimidin-5-yl)methyl][(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
1-[4-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
3-[4-(3-chloro-4-fluorophenyl)piperazine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
4-{4-[(1-ethenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-2-methyl-6-propylpyrimidine
(3aS,6aS)-2-[5-(4-methoxyphenyl)furan-2-carbonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-7-oxo-N-[2-(thiophen-2-yl)ethyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
3-amino-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
N-(2-methoxyethyl)-N,1-dimethyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 4-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}piperidine-1-carboxylate
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
5-acetyl-2,4-dimethyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrrole-3-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
3-fluoro-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]benzonitrile
8-(isoquinolin-1-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-4-[5-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)furan-2-yl]but-3-yn-2-ol
N,2,7-trimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
ethyl 2-{1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]piperidin-2-yl}acetate
4-(2-oxo-1-phenylpyrrolidine-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4,6-dimethylpyrimidine
7-(2-methylphenyl)-4-(1,3-thiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-fluoro-3-({[(2-methoxyphenyl)methyl]amino}methyl)-1-(oxolan-2-ylmethyl)-1,2-dihydroquinolin-2-one
7-methyl-2-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
(2S)-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)butan-1-ol
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-[methyl(piperidin-4-yl)amino]acetamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-(3-fluorophenyl)pyridine-3-carboxamide
4-[(5-chloro-3-methyl-1-benzothiophen-2-yl)sulfonyl]piperazine-2-carboxylic acid
1-(2-methoxy-5-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
11-[(pyridin-3-ylmethyl)amino]-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)-1,4-diazepan-5-one
8-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-({[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}amino)pyridine-4-carbonitrile
N-[2-(pent-4-enoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-4-(trifluoromethyl)benzamide
3-{[(5-methylthiophen-2-yl)methyl]({[1-(propan-2-yl)piperidin-4-yl]methyl})amino}propan-1-ol
(4aS,8aR)-1-(3-hydroxypropyl)-6-{imidazo[1,2-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
2-chloro-N,N-dimethyl-5-[({2-[(2R)-pyrrolidin-2-yl]ethyl}carbamoyl)amino]benzamide
2-(adamantan-1-yl)-1-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one