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4-(4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
2-(4-chlorophenyl)-4-[3-(1H-1,2,4-triazol-3-yl)benzoyl]morpholine
2-[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]-1H-1,3-benzodiazole-5-carbonitrile
4-{[2-(difluoromethoxy)phenyl]methyl}-2-methyl-1,4-oxazepane
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)pent-4-enamide
1-{2-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
3-[5-(2-carbamoylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(propan-2-yl)propanamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-3,4,7-trimethyl-1H-indole-2-carboxamide
(1R,7S)-N-ethyl-N-methyl-3-[2-(4-methylphenyl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-{4-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carbonyl]phenyl}-2-methylbutan-2-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-cyclobutanecarbonylpyrrolidin-3-yl]methanol
methyl 2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
1-(ethanesulfonyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-(hydroxymethyl)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}cyclopropane-1-carboxamide
1-methyl-N-[(3-methylphenyl)methyl]-6-oxo-N-(oxolan-2-ylmethyl)-1,6-dihydropyridine-3-carboxamide
N-[(4-acetamidophenyl)methyl]-2-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]acetamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(6-methoxypyridazin-3-yl)-1H-pyrazol-1-yl]acetamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(2-oxopyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-{[(furan-3-ylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
1-[(4-chlorophenyl)methyl]-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
4-[1-(pyrrolidin-1-yl)ethyl]-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine
N-methyl-4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
3-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}propane-1,2-diol
1-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-6-carboxamide
4-(3-hydroxypyridine-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(2-amino-1,3-thiazol-4-yl)propan-1-one
2-(1H-imidazol-2-yl)-N-[2-(4-sulfamoylphenyl)ethyl]benzamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
2-amino-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-methylpropan-1-one
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-(pent-4-enamidomethyl)benzoate
4-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-(1-methyl-1H-pyrazol-3-yl)-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
2-ethyl-8-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-[4-(2-cyclohexyl-1H-imidazol-1-yl)phenyl]-5-methyl-4H-1,2,4-triazole
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pentan-1-one
N-[(3S,4R)-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-3-ethylpiperazin-2-one
1-[2-(dimethylamino)-4-{[2-(5-methylthiophen-2-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-(1-cyclohexylpiperidin-3-yl)-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-5-(phenoxymethyl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-methyl-2-(pyrrolidin-1-yl)propan-1-one
2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-N,4-dimethylaniline
4-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}benzene-1-sulfonamide
(1r,4r)-4-{[1-(4,6-dimethylquinazolin-2-yl)piperidin-4-yl]amino}cyclohexan-1-ol