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1-cyclobutanecarbonyl-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
1-(2-{1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-[2-(azepan-1-yl)-2-phenylethyl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
2-{9-[(4-cyanophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)pyrazine-2-carboxamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-[(4-methylphenyl)sulfanyl]piperidine-1-carboxamide
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-4-(2-methylphenyl)piperazine
2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(4-methyl-1,3-thiazole-5-carbonyl)-8-azabicyclo[3.2.1]octane
5-[2-(benzyloxy)phenyl]-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,1-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
5-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}-2-(furan-2-yl)pyrimidine
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amino}acetamide
ethyl({imidazo[1,2-a]pyrimidin-6-ylmethyl}){[2-(prop-2-en-1-yloxy)phenyl]methyl}amine
(4aS,8aR)-6-(2-fluorobenzenesulfonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
2-[(1-cyclopentanecarbonylpiperidin-4-yl)formamido]-2-(2-fluorophenyl)acetic acid
6-fluoro-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)urea
2-{4-[(5-ethylfuran-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(dimethyl-1,2-oxazol-4-yl)-N-(4-phenyl-1,2,3-thiadiazol-5-yl)pyrrolidine-1-carboxamide
2-[5-(1H-imidazol-4-ylmethyl)-3-(oxan-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-5-methylpyrimidine
[1-(3-{1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenyl)ethyl]dimethylamine
(1R,3S)-7-[2-(benzyloxy)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
3-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]azetidin-3-yl}pyridine
4-methyl-2-(4-methylpiperazin-1-yl)-N-[(2R)-pyrrolidin-2-ylmethyl]pyrimidine-5-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole
2-amino-6-(3-hydroxyphenyl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
6-fluoro-2-[({[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]quinolin-4-ol
N-(1-benzylpiperidin-4-yl)-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-1-(2-methoxyphenyl)-N-methylpiperidin-4-amine
3-(2-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
[(2S,4R)-4-(dimethylamino)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-2-yl]methanol
3-(1,4-diazepane-1-carbonyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzene-1-sulfonamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
3-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-4-fluorobenzene-1-sulfonamide
N-[(3S,4R)-1-(1,3-benzoxazol-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(thiophen-2-yl)propanoyl]piperidin-3-yl]propanoic acid
3-chloro-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-hydroxybenzamide
4-cyano-1-methyl-N-[2-oxo-2-(piperazin-1-yl)ethyl]-1H-pyrrole-2-carboxamide
4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-cyclohexyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(prop-2-yn-1-yl)acetamide
3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}-1-[2-(trifluoromethoxy)benzenesulfonyl]piperidine
N-(2-{[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]amino}ethyl)acetamide
4-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-N,N-dimethyl-4-oxobutanamide
4-{3-cyclopropyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
8-(1H-imidazol-2-ylmethyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{2-[(4-{[(4-methylphenyl)amino]methyl}phenyl)formamido]ethyl}acetamide