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2-ethoxy-5-[2-(pyrimidin-2-yl)pyrimidin-4-yl]benzoic acid
N,N-dimethyl-7-(4-methylpyridine-3-carbonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1-methyl-1H-pyrrol-3-yl)acetamide
{1-methyl-5-[(8-methylquinolin-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
2-(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)-N-[(4-acetamidophenyl)methyl]acetamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
6-fluoro-2-{[4-(2,2,2-trifluoroethyl)piperazin-1-yl]methyl}quinolin-4-ol
N-cyclopropyl-N-(pyridin-3-ylmethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-(2-methylphenyl)-4-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
[3-(1H-imidazol-1-yl)propyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
9-[2-amino-6-(methylamino)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-hydroxy-4-methylazepan-1-yl)-4-(4-methoxyphenyl)butane-1,4-dione
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
N4-ethyl-N2-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
5-butyl-4-methyl-6-{4-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
3-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]pyridin-2-ol
2-{4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]morpholin-3-yl}acetic acid
1-[(4-chlorophenyl)methyl]-N-[(4-ethylphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
({5-[1-(1-benzothiophene-2-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-benzoyl-1-[2-(2-methoxyphenoxy)ethyl]piperidine
1-{2-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1-{[1-(1H-indole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(5-{[2-(benzylamino)pyrimidin-5-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
6-methyl-2-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyridine-3-carbonitrile
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-3-(3-methylphenoxy)azetidine
4-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,3-oxazole-5-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(6-methyl-2-phenylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
N-(4-chlorophenyl)-5-[4-hydroxy-1-(thiophen-2-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
(1R,9S)-5-amino-12-methyl-3-(6-methyl-1H-indol-3-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
(1S,6R)-N-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-[2-methoxy-5-({[3-(pyridin-3-yl)propyl]carbamoyl}amino)phenyl]propanamide
N-(2-hydroxyethyl)-3-(4-methylphenyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-5-carboxamide
4-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1,3-thiazol-2-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-({2-[(furan-2-ylmethyl)(pyridin-2-ylmethyl)carbamoyl]phenyl}amino)acetic acid
3-[(3R,4S)-1-[(2-chloro-6-methylphenyl)carbamoyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-{[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(cyclopentylcarbamoyl)pyrrolidine-3-carboxylic acid
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(pyrrolidin-3-yl)benzamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(5-methylpyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-[3-chloro-4-(dimethylcarbamoyl)phenyl]-4-ethoxypiperidine-1-carboxamide
N-butyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
5-fluoro-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-2-amine