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6-[4-fluoro-3-(hydroxymethyl)phenyl]-3,4-dihydroquinazolin-4-one
2-(dimethylamino)-N-{[1-(ethoxymethyl)cyclopropyl]methyl}-2-(3-methylphenyl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
4-[(7-hydroxyquinolin-3-yl)methyl]piperazine-2-carboxylic acid
1-(2-hydroxy-3-{2-methoxy-4-[(4-methylpiperidin-1-yl)methyl]phenoxy}propyl)piperidin-4-ol
2-(4-chlorophenyl)-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
9-(2-methoxyethyl)-N,N,1-trimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-sulfonamide
[(3S,5R)-1-(1H-indole-5-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
methyl 5-[(1-propyl-1H-1,3-benzodiazol-5-yl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-cyclooctyl-2-{[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}acetamide
1-(4-fluorophenyl)-4-[2-(methylsulfanyl)benzoyl]-1,4-diazepane
N-[2-(morpholin-4-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}propanoic acid
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-ol
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidin-3-ol
4-ethyl-3-(1-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2,6-dimethyl-4-(4-phenyl-1,4-diazepane-1-carbonyl)quinoline
3-(1H-imidazol-1-ylmethyl)-N-(2-methyl-5-sulfamoylphenyl)piperidine-1-carboxamide
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
3-({[2-(2H-1,3-benzodioxol-5-yl)ethyl]amino}methyl)piperidin-3-ol
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]acetamide
{2-ethoxy-5-[4-phenyl-1-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-imidazol-5-yl]phenyl}methanol
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
5-(4-amino-5-methylpyrimidin-2-yl)-N-(2-hydroxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(benzylsulfamoyl)[3-(4-methyl-1,3-thiazol-5-yl)propyl]amine
2-[4-(1-benzofuran-2-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethan-1-amine
2-(4-{[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}piperidin-1-yl)acetamide
5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-methoxypyrimidine
(4aR,7aS)-1-(2-methylpropanoyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
6-[4-(2-phenylethyl)piperidine-1-carbonyl]piperazin-2-one
1-phenyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
2-{2-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
2-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[5-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
1-(cyclohex-3-en-1-ylmethyl)-3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]piperidine
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-1-(2-methoxyphenyl)-1H-pyrazole
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-[(3S)-3-acetamidopyrrolidin-1-yl]propanamide
2-methyl-5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,4-dihydropyridin-4-one
N-[(3S)-1-benzylpiperidin-3-yl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
(4aR,7aS)-1-(2-methylpropyl)-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(6-ethyl-2-methylquinoline-4-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-cyclobutyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
3-(5-methanesulfonamido-2-methylphenyl)-1-[2-(piperidin-1-yl)ethyl]urea
4-[(diethylamino)methyl]-5-ethyl-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]furan-2-carboxamide
4-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-4-oxobutanamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide