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5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
5-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}-1-ethyl-1H-1,2,4-triazole
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
N-methyl-N-[1-(pyridin-3-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(dimethylamino)-N-[2-methyl-2-(4-methylpiperazin-1-yl)propyl]-2-(3-methylphenyl)acetamide
3-[(2,2-dimethylmorpholin-4-yl)sulfonyl]-N-(oxolan-3-ylmethyl)benzamide
ethyl 1-[(6-methylpyridin-2-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
2,8-dimethyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(6-fluoroquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(oxan-2-yl)ethyl]propanamide
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-(propan-2-yl)pyrrolidin-2-one
1-(oxan-4-yl)-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepane-6-carboxylic acid
1-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-5,5-diphenylpiperidin-2-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
2-({[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
2,2-difluoro-N-[(1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
2-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]benzonitrile
4-[2-(2-ethylphenoxy)ethyl]-1,4-oxazepan-6-ol
3-[(4aR,7aS)-4-[(4-methyl-1,3-thiazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
4-fluoro-N-(2-methoxyethyl)-3-methyl-N-(thiophen-2-ylmethyl)benzamide
6-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3,4-difluorophenyl)methyl]-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2,6-dimethylphenoxy)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}azetidine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(1H-pyrazol-5-yl)furan-2-sulfonamide
2-(3-hydroxyphenyl)-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
{1-methyl-5-[4-(piperidin-1-ylmethyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
2-[2-(furan-2-yl)phenyl]-1-(thiolan-3-yl)-1H-imidazole
1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
methyl 1-({4-[4-(thiophen-2-yl)butanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]thian-4-amine
1-methyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-(azocane-1-carbonyl)-N-(oxan-3-yl)benzene-1-sulfonamide
1-(2-hydroxyethyl)-5-[(2-phenyl-1,3-thiazol-5-yl)methyl]-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridin-2-ol
8-{[4-(3-ethylmorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
(1S,5R)-3-benzyl-6-(2-methoxy-5-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1'-[5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]spiro[indene-1,4'-piperidine]
2-[3-({[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]amino}methyl)piperidin-1-yl]ethan-1-ol
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}furan-3-carboxamide
N-[1-(pyrazin-2-yl)propan-2-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
methyl N-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}carbamate
3,5-difluoro-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyridine-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]urea
4-ethyl-2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-methylpyrimidine
1-cyclopropyl-4-({[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}methyl)pyrrolidin-2-one
3-methyl-3-[2-(2-oxopiperidin-1-yl)ethyl]-1-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
4-{1-[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]ethyl}-2-methyl-1,3-thiazole