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2-(methylsulfanyl)-N-[(3R,4S)-4-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl]acetamide
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
(3S,4S)-1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
3-methoxy-N-[2-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
(1S,6R)-9-(6-methyl-2-propylpyrimidin-4-yl)-3,9-diazabicyclo[4.2.1]nonane
2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}-2-phenylacetic acid
ethyl[(5-fluoro-3-methyl-1H-indol-2-yl)methyl][(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyridine-4-carboxamide
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-2-methoxyacetamide
1-(4-ethylpiperazin-1-yl)-3-{3-[(4-fluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol
1-(4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-N-(pyridin-3-yl)benzamide
N-(3-chloro-4-methoxyphenyl)-6-{2-[4-(methylsulfanyl)phenyl]acetyl}-6-azaspiro[2.5]octane-1-carboxamide
N-(3-methoxyphenyl)-2-{4-[2-(pyridin-4-yl)acetyl]morpholin-3-yl}acetamide
11-{[(5-fluoro-2-methylphenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
{imidazo[1,2-a]pyrimidin-2-ylmethyl}({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[4-(furan-2-yl)benzoyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
({3-[1-(dimethylamino)ethyl]phenyl}methyl)(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-{1-[3-(diethylamino)pyrrolidin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
2-(4-chloro-2-methylphenoxy)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}acetamide
9-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
N-[1-(4-methylphenyl)ethyl]-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}acetamide
N-[(4-hydroxy-3-methoxyphenyl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(quinolin-5-ylmethyl)amine
3-{2-oxo-2-[3-(4-propylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1,3-oxazolidin-2-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{2-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
[1-phenylmethanesulfonyl-4-(3-phenylpropyl)piperidin-4-yl]methanol
3-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[1-(3-methylpyridin-2-yl)propyl]urea
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](1H-imidazol-4-ylmethyl)amine
1-(cyclohexylmethyl)-5-[(2-hydroxyethyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
2-amino-6-cyclobutyl-4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyridine-3-carbonitrile
methyl 2-(cyclopropylsulfamoyl)-6-(3,5-dimethylbenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)propanamide
N-[2-(3-propoxyphenyl)ethyl]spiro[2.2]pentane-1-carboxamide
3-(3-phenoxyazetidine-1-carbonyl)piperidine-1-carboxamide
4-(4-methoxyphenoxy)-1-(2-methylfuran-3-carbonyl)piperidine
(2S,4S)-N-ethyl-4-[2-(2-hydroxyphenyl)acetamido]-1-(3-methoxypropanoyl)pyrrolidine-2-carboxamide
5-(2-chlorophenyl)-N-[2-(4-hydroxypiperidin-1-yl)ethyl]furan-2-carboxamide
2-benzyl-N-[(4-phenyloxan-4-yl)methyl]-1,3-thiazole-4-carboxamide
1-[(3-chloropyridin-4-yl)methyl]-4-[(dimethylamino)methyl]piperidin-4-ol
1-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-methyl-6-(propan-2-yl)pyrimidin-4-amine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(4aR,8aS)-6-{[3-(4-chlorophenoxy)phenyl]methyl}-1-(2-methoxyethyl)-decahydro-1,6-naphthyridin-2-one
1-ethyl-3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
6-[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-2-carbonitrile
N-methyl-1-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
[4-(6-methyl-2-phenylpyrimidin-4-yl)morpholin-2-yl]methanamine