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(2S,4R)-4-[4-(4-chlorobenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
dimethyl[(2-{[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methyl]amine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-(pyrazin-2-yl)propanamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}acetamide
(1S,5R)-6-cyclobutanecarbonyl-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyridin-2-ylmethyl)amine
2-ethyl-4-phenyl-9-(1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]pyrimidine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-methyl-2-(phenylamino)propanamide
6-(1H-1,2,4-triazol-1-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-ethyl-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
4-[(3-fluoro-4-methoxyphenyl)methyl]-1-phenylpiperazin-2-one
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-[(8-methoxyquinolin-5-yl)methyl]-1-methylurea
2-(5-chloro-2-ethoxyphenyl)-N,N-dimethylpyridine-3-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-2-carbonyl)piperidine
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5,6-dimethylpyrimidine
2-[(1S,5R)-6-[3-(dimethylamino)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-cyclopropyl-1,3-oxazole-4-carboxamide
N3-[3-(dimethylamino)-2,2-dimethylpropyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
6-methyl-2-[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
(4aS,7aR)-1-(4-hydroxy-3-methoxybenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2,6-dimethoxypyridine-3-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]propan-1-one
3-[(2R,3R,6R)-5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-{3-[4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl]propyl}morpholine
5-ethyl-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
[1-(2-methoxy-5-methylbenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
2-(2-methylfuran-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
(3aS,6aS)-2-methyl-5-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(2-phenoxyethyl)amine
3-[4-(piperidine-1-carbonyl)phenyl]-1-[1-(pyridin-4-yl)propan-2-yl]urea
(3aS,6aR)-5-[2-(1H-indol-3-yl)ethyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-{[1-(phenylcarbamoyl)pyrrolidin-3-yl]methyl}benzoic acid
4-(1-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
4-(hydroxymethyl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]azepan-4-ol
(2S,3R)-2-[2-(6-ethoxyquinolin-2-yl)-1H-imidazol-1-yl]-3-hydroxybutanamide
(3R,4R)-4-(azepan-1-yl)-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
8-chloro-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}quinoline-2-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
3-amino-N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
3-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
(3S)-1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidin-3-ol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-5-methyl-1H-indazole-3-carboxamide
3-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
1-(2-chlorobenzoyl)-4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
2,6-dimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]quinoline-4-carboxamide