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N-[1-(dimethylamino)propan-2-yl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-[({5-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-6-methoxypyrimidin-4-amine
5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
(2H-1,3-benzodioxol-5-ylmethyl)[(2-methyl-1H-imidazol-4-yl)methyl][(4-methylphenyl)methyl]amine
2-(2,3-dihydro-1H-inden-1-yl)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]acetamide
1-{3-[(3R)-3-cyclopropyl-3-hydroxy-4,4-dimethylpyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
5-cyclopropyl-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,3,4-oxadiazol-2-amine
(1R,7S)-3-cycloheptyl-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
6-methyl-5-[5-(oxan-4-yl)-1,2,4-oxadiazol-3-yl]-2-(pyrazin-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-cyclopentyl-1-methyl-5-(naphthalen-1-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[3-(1H-indol-1-yl)propyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
2,4-dichloro-3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)phenol
3-(piperidin-3-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)benzamide
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
methyl 2-[8-(2H-1,3-benzodioxol-5-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
3-methyl-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
N,2-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,3-thiazole-4-carboxamide
N-[2-(morpholin-4-ylmethyl)phenyl]-3-(propoxymethyl)pyrrolidine-1-carboxamide
1-[3-tert-butyl-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-3-methylbutan-1-ol
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(3-methoxyphenyl)propan-1-one
1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-[4-(4-ethoxy-3-methylphenyl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(4-hydroxyazepan-4-yl)methyl]-4-methyl-5-phenylthiophene-2-carboxamide
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-(2-methoxyphenoxy)-2-methylpropan-1-one
7-fluoro-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline
2-methoxy-4-(8-methoxy-2-methylquinolin-5-yl)pyridine-3-carbonitrile
3-(5-{[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,4-triazol-3-yl)pyridine
N-[2-(dimethylamino)ethyl]-8-fluoro-N-(oxolan-2-ylmethyl)quinoline-2-carboxamide
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(thiophene-2-carbonyl)pyrrolidine-2-carboxamide
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)morpholine
N-(3-methoxypropyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-benzyl-N-ethyl-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[(1-ethyl-1H-pyrazol-4-yl)methyl][1-(morpholin-4-yl)propan-2-yl]amine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-phenylmethanesulfonylpiperidine
8-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(2S)-1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidine-2-carbonyl]morpholine
5-(8-methoxy-2-methylquinolin-5-yl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-hydroxyethyl)-8-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-cyclopentyl-1-methyl-5-[4-(piperidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(carbamoylmethyl)-2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
1-{pyrazolo[1,5-a]pyridine-7-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
(1R,3S,5S)-8-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
[(3S,5R)-5-(morpholin-4-ylmethyl)-1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]methanol
3-(3-chloro-4-methoxyphenyl)-1H-1,2,4-triazole-5-carboxamide
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1,2-oxazole
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-(2-hydroxypyridin-3-yl)urea
(2S)-N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide