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1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}piperidin-2-one
(4aS,7aR)-1-[(2-ethylphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{4-[1-(5-fluoro-2-methylphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-methylfuran-2-yl)methyl]acetamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
(2-chloro-6-fluorophenyl)(4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
2-{[4-(2-hydroxyethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(6-methylpyridazin-3-yl)-4-phenoxypiperidine-4-carboxylic acid
N'-(2,4-dimethylphenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanediamide
2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)thiomorpholine
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[4-(4-methylphenyl)benzoyl]piperidine
3-{[(cyclohexylmethyl)amino]methyl}-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
[(3R,4R)-1-(3,5-dimethoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(4aR,8aR)-7-(5-ethyl-1H-pyrrole-2-carbonyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
N-methyl-N-[2-(morpholin-4-yl)propyl]-2-(phenylamino)pyrimidine-5-carboxamide
4-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2,6-dimethylphenyl acetate
2-methyl-4-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyridine
7-(cyclobutylmethyl)-2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(4aS,7aR)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-(4-methoxy-2-methylbenzoyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine
N-[3-(6-methoxypyridin-3-yl)phenyl]acetamide
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-5-methyl-1,2-oxazole-3-carboxamide
2-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
1-cyclopentyl-4-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]piperazin-2-one
4-{2-[(3-hydroxypiperidin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-methoxypyridine-3-carbonitrile
1-(1-methyl-1H-imidazole-5-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)propanamide
2-(pyridin-3-ylmethyl)-9-[2-(pyrrolidin-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[({[2-(azocan-1-yl)pyridin-3-yl]methyl}amino)methyl]thiophen-2-yl}ethan-1-one
1-(1,2,4-oxadiazol-3-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-{4-[(3-hydroxyphenyl)methyl]piperazin-1-yl}-2-(pyrrolidin-3-yl)ethan-1-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(dimethylsulfamoyl)piperidin-3-yl]propanamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
2-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-(2-methoxyethyl)-1-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
butyl 7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate
3-[(1-benzylpiperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
1-ethyl-5-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
4-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
(3R,5S)-N-[2-(1H-indol-1-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-[1-(2,3-dihydro-1H-inden-4-yl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl]acetamide
5-[(2-propyl-1H-imidazol-1-yl)methyl]-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-5-methoxy-1H-indazole
1-{3-[(dimethylamino)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
3-[(3R,4S)-1-(3-fluoropyridin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-{1-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}benzoic acid