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N-(1-hydroxy-2-methylpropan-2-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
methyl 3-[(2-methylpropanamido)methyl]-5-[3-(trifluoromethyl)benzamido]benzoate
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
2-(4-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-(3-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}-4-methoxyphenyl)acetic acid
1-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1H-indole-6-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{1-[1-(4-hydroxybutyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
4-[7-(3-chloro-4-fluorobenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1-[(3-ethoxy-4-methoxyphenyl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(3-phenyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
N,1-dimethyl-3-(propan-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
N-[(3-methyloxetan-3-yl)methyl]-4-(methylsulfanyl)benzamide
(1S,5R)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-benzyl-3-methyl-4-[2-(methylsulfanyl)ethyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decane
1-[5-cyclobutyl-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-phenyl-1,2,4-triazin-3-amine
2-(2-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-[(3-fluorophenyl)methyl]-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-methoxy-3-{[4-(propan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
2-(4-{[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]methyl}cyclohexyl)-1H-1,3-benzodiazole
(1S,5R)-6-benzyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-methoxyethyl)-8-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
2-chloro-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-5-(trifluoromethyl)benzamide
N-methyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
(1r,4r)-4-{[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]methyl}cyclohexane-1-carboxylic acid
1-benzyl-N-(oxan-4-yl)-1H-pyrazol-5-amine
4-({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)-1,4-diazepan-2-one
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1,2-dimethyl-4-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperazine
1-[(3-fluorophenyl)methyl]-4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1,4-diazepane
4-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
3-methyl-1-(4-{[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)but-2-en-1-one
3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[4-methyl-3-(propan-2-yl)phenyl]urea
2-{[methyl({[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]benzonitrile
ethyl 2-chloro-5-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}benzoate
6-[4-(acetamidomethyl)piperidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
2-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}sulfonyl)benzonitrile
2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}acetamide
1-cyclohexyl-N3-[1-(6-methoxynaphthalen-2-yl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(phenylsulfanyl)ethyl]benzamide