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2-[4-(3-chloropyridin-2-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-[(dimethylamino)methyl]-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]azepan-4-ol
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
2-{[4-(4-aminopyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
4-({2-[1-(2-fluoro-4-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-yl)ethan-1-ol
4-(piperidin-1-ylmethyl)-N-[3-(pyridin-2-yl)propyl]benzamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-(2-phenyl-1H-imidazole-4-carbonyl)piperidin-3-ol
[1-(2-methoxyphenyl)ethyl](methyl)(piperidin-4-ylmethyl)amine
8-methoxy-3-(pyridin-3-ylmethyl)-3,4-dihydroquinazolin-4-one
2-cycloheptyl-1-[4-({4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]ethan-1-one
N1-(pyridin-3-yl)-N2-[4-(pyridin-3-yl)pyrimidin-2-yl]ethane-1,2-diamine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-N'-(2-methylphenyl)propanediamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
(3aR,5S,6S,7aS)-2-[(3R)-3-hydroxy-3-phenylpropyl]-octahydro-1H-isoindole-5,6-diol
(1S,5R)-6-(morpholine-4-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-N-methyl-3-(4-methylpiperazine-1-carbonyl)-N-(naphthalen-1-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(2-methylpropyl)benzoyl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-ol
5-benzyl-4-(2-methoxyacetyl)-1-(4-methylphenyl)piperazin-2-one
3-(3-methylbutyl)-1-{[4-(methylcarbamoyl)phenyl]methyl}-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-[(3-methoxyphenyl)amino]-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]butanamide
1-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
2-methoxy-N-({7-[2-(4-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-phenylacetamide
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2,1-benzoxazole-3-carboxamide
N-(furan-2-ylmethyl)-6-methoxy-2-oxo-N-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-3-pentanamidobenzamide
N,N-dimethyl-3-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}sulfamoyl)benzamide
2-[4-(4-fluorophenyl)-2-[(3-oxopiperazin-1-yl)methyl]phenoxy]acetic acid
1-{2-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrimidin-4-yl}pyrrolidin-3-ol
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
(1R,5R)-N,N-dimethyl-6-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-methyl-6-[3-(propan-2-yl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
2-(2-hydroxyethyl)-9-[(6-methylquinolin-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N3-cycloheptyl-4-oxo-1-(propan-2-yl)-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3aS,6aS)-2-[(5-methylpyrazin-2-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[4-(2-methylfuran-3-carbonyl)-1,4-oxazepan-6-yl]methanol
7-fluoro-2-methyl-4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}quinoline
N-methyl-N-(propan-2-yl)-2-(pyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}benzoic acid
N-(3,4-dimethylphenyl)-2-({[(2S)-5-oxopyrrolidin-2-yl]methyl}(pyridin-4-ylmethyl)amino)acetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(2-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-methoxyethyl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-(2-phenoxyethyl)-1-(quinolin-2-ylmethyl)piperidine-4-carboxylate
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,3-dimethoxybenzamide
6-(methoxymethyl)-1-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(3-chlorophenyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol