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4-(1H-imidazole-4-carbonyl)-2-(naphthalen-1-ylmethyl)morpholine
4-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-(furan-2-ylmethyl)-4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)piperidine
1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazole
1-{2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-ethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(propan-2-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[(4aS,7aR)-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]cyclopropane-1-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-5-cyclopropyl-1,2-oxazole-3-carboxamide
9-methyl-6-(1,2,3,4-tetrahydroisoquinolin-5-yl)-2,3,4,9-tetrahydro-1H-carbazol-1-one
1-[(4aR,8aR)-7-{[2-(cyclopentyloxy)phenyl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
1-(2-ethoxyphenyl)-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
(3aS,6aS)-2-methyl-5-[4-(piperidin-1-ylmethyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(S)-carbamoyl(phenyl)methyl]propanamide
5-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2-(propan-2-yloxy)-N-(pyridin-4-ylmethyl)acetamide
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-3-methylthiophene-2-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-(1-benzylpyrrolidin-3-yl)-3-{1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}propanamide
5-(oxolan-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}thiophene-2-carboxamide
[(3R,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-ethoxy-5-[2-(4-phenylpiperazin-1-yl)pyrimidin-4-yl]benzoic acid
methyl 3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})amine
N-[2-(1H-imidazol-4-yl)ethyl]-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamide
[3-(8-methoxyquinolin-5-yl)-1H-1,2,4-triazol-5-yl]methanol
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-1-yl]pyridine-4-carboxamide
4-(2-{[(3-methylthiophen-2-yl)methyl]amino}benzoyl)piperazin-2-one
2-{4-[1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
2-(1-cyclopentyl-4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(2-methanesulfonylethyl)piperazine
3-(3-hydroxy-1,2-oxazol-5-yl)-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]naphthalen-1-ol
2-[(1H-imidazol-2-ylmethyl)(methyl)amino]-2-(3-methoxyphenyl)acetic acid
2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-methylpyridine-3-carbonitrile
methyl 3-benzamido-1-(oxolan-2-ylmethyl)-5-{[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-benzyl-4-{[4-(difluoromethoxy)phenyl]methyl}-1,4-diazepan-6-ol
2-(2,4-dichlorophenoxy)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
3-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-N-methylpropanamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(3-ethoxy-2-hydroxypropyl)amine
4-(hydroxymethyl)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-ol
4-cyano-N-(furan-2-ylmethyl)-1-methyl-N-(pyridin-4-ylmethyl)-1H-pyrrole-2-carboxamide
2-[3-(4-fluorophenyl)pyrrolidin-1-yl]pyrimidin-4-amine
8-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-oxa-8-azaspiro[4.6]undecane
4-{5-methyl-3-[(phenylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
N-benzyl-4-cyano-1-methyl-N-[(3-methylpyridin-2-yl)methyl]-1H-pyrrole-2-carboxamide
1-[4-(4-methyl-1,4-diazepan-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one