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1-[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}thiophen-3-yl)methyl]pyrrolidine
1-(2-ethoxyethyl)-N,3-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-pyrazole-5-carboxamide
dimethyl[(2-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}phenyl)methyl]amine
ethyl 2-(1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperidin-2-yl)acetate
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-methyl-5-propyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,2-dihydroquinolin-2-one
5-{[(1H-imidazol-2-ylmethyl)(propan-2-yl)amino]methyl}pyrrolidin-2-one
prop-2-en-1-yl 3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
8-chloro-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}quinoline
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
5-(methoxymethyl)-N-[2-(N-methylmethanesulfonamido)ethyl]furan-2-carboxamide
6-[(diethylamino)methyl]-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[1-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
3-{[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
(4aR,8aR)-2-methanesulfonyl-7-(4-phenoxybutyl)-decahydro-2,7-naphthyridin-4a-ol
(3S,5R)-N3-cyclopropyl-N5-(2,3-dihydro-1H-inden-5-yl)piperidine-3,5-dicarboxamide
2-amino-1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
[(1-ethyl-1H-imidazol-2-yl)methyl][(8-methoxyquinolin-2-yl)methyl]methylamine
(2S,4S)-4-amino-1-(3-cyano-5-fluorobenzoyl)-N-ethylpyrrolidine-2-carboxamide
N-benzyl-N-methyl-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
1-(5-methyl-1,3-oxazole-4-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
2-(1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
5-(oxan-4-yl)-3-(1-phenylcyclopropyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
5-{[(1R,5S,6S)-6-(cyclopentylcarbamoyl)-3-azabicyclo[3.1.0]hexan-3-yl]methyl}-2-hydroxybenzoic acid
1-cyclohexyl-N3-methyl-4-oxo-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[(2,4-dimethoxyphenyl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(4aS,7aR)-1-[(3-methylthiophen-2-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-hydroxypropyl)-9-(4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[4-(2-aminopyridin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
6-[1-(4-fluorophenyl)cyclopropanecarbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
1-ethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(1H-imidazol-1-ylmethyl)-1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-ol
2-[4-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
9-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
1-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(2R)-2-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(2,6-dimethylpyridin-4-yl)piperazine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-N-(pyrazin-2-ylmethyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)-3-methylpyrazine
N,1-bis(furan-2-ylmethyl)-N-(prop-2-en-1-yl)piperidine-4-carboxamide
1-(2-methyloxolane-2-carbonyl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
4-[2-(2-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}phenoxy)ethyl]morpholine
2-{3-[(2S,4R,6R)-6-cyclohexyl-4-acetamidooxan-2-yl]phenoxy}acetamide
2-[(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole