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4-(2,6-dimethylpyridin-3-yl)-2-(1H-pyrazol-4-yl)pyrimidine
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-imidazole
1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
7-[(3-methoxyphenyl)methyl]-6-oxo-N-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(1,4-oxazepan-4-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
4-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-N-(2-hydroxyethyl)pyridine-2-carboxamide
ethyl 4-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperazine-1-carboxylate
4-(hydroxymethyl)-1-(3-methoxypyrazin-2-yl)piperidin-4-ol
2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-[(pyridin-3-ylmethyl)amino]benzamide
2-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[(4aR,7aS)-6,6-dioxo-4-(3-phenoxypropyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
2-(3-chlorophenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
2-(4-{[4-(cyclohex-3-en-1-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
1-[4-(1H-imidazol-1-yl)benzamido]cycloheptane-1-carboxamide
3-{1-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
3-chloro-5-[3-(2-methylphenyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(adamantan-2-yl)-6-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[5-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyridin-3-yl)propanamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[methyl(phenyl)amino]propyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
{5-[2-(2-butyl-5-chloro-1H-imidazol-4-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-2-yl}methanol
1-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}piperidine-4-carboxamide
1-[(3-fluorophenyl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
(1R,3R,5S)-3-(4-methoxyphenyl)-8-[(2R)-oxolane-2-carbonyl]-8-azabicyclo[3.2.1]octane
2-{4-[1-(oxan-4-yl)piperidine-4-carbonyl]piperazin-1-yl}pyrimidine
4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-fluoro-2-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)quinoline
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(2-methylpropanoyl)piperidin-4-yl]propanamide
5-{[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
{4-[(3-fluorophenyl)methyl]-1-(thiophene-2-sulfonyl)piperidin-4-yl}methanol
1-ethyl-N-(1-methylpiperidin-4-yl)-3-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(6-methyl-2-propylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
2-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)pyridine-3-carboxylic acid
2-(cyclopropylmethyl)-8-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
6-chloro-8-methyl-3-(morpholin-2-ylmethyl)-3,4-dihydroquinazolin-4-one
{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]pyridin-4-yl}methanol
(2-{[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)dimethylamine
1-(3,4-dimethoxyphenyl)-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
3-(3-hydroxyquinoxalin-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
N-cyclopropyl-5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(5-ethyl-1-benzofuran-3-yl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}acetamide
1-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(2-methanesulfonylethyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
2-{4-[1-(2-methylpropyl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
9-[2-(3,4-dimethylphenoxy)ethyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one