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3-cyclopropyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-phenyl-1H-1,2,4-triazole
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}ethane-1-sulfonamide
N-(3-chloro-4-fluorophenyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
2-[4-cyclobutyl-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-cyclopropyl-5-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]pyrrolidine-3-carboxamide
methyl 6-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-[(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-butanamido-N-[1-(dimethylamino)propan-2-yl]benzamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
2-amino-N,3-diethyl-N-[(5-methylfuran-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}acetamide
8-[(5-ethylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2E)-1-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
7-(dimethylamino)-4-[2-(3-methylphenyl)pyrimidin-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
3-(3-{1-[(2R)-2-hydroxy-2-phenylethyl]-1H-pyrazol-3-yl}phenyl)pyrazine-2-carbonitrile
8-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N6-cyclopropyl-N4-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N4-methylpyrimidine-2,4,6-triamine
1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{[5-(furan-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-methanesulfonylpiperazine
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
4-[3-(2-hydroxyphenyl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-fluoro-5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(1S,9R)-11-{2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
6-[1-(2-methyl-1,3-benzoxazole-6-carbonyl)piperidin-3-yl]pyrimidin-4-ol
4-ethyl-3-{1-[5-(methanesulfonylmethyl)pyridin-2-yl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-dimethyl-2-{[3-(trimethyl-1H-pyrazol-1-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-[2-(2,3-dihydro-1H-inden-1-yl)acetamido]cyclopentane-1-carboxylic acid
methyl[(4-methyl-1H-imidazol-5-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
(5R)-5-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-3-({methyl[1-(methylcarbamoyl)propan-2-yl]amino}methyl)benzamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1,3-oxazole-4-carboxamide
2-[(dimethylcarbamoyl)amino]-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
3-[4-(2-oxopyrrolidin-1-yl)phenyl]-1-{3-[(pyridin-3-yl)amino]propyl}urea
5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-(ethylsulfanyl)pyrimidine
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-4-(piperidin-3-yl)benzamide
4-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
1-[4-phenyl-1-(quinoline-6-carbonyl)piperidin-4-yl]ethan-1-one
2-[(1-acetylpiperidin-4-yl)(methyl)amino]-1-(4-hydroxyphenyl)ethan-1-one
[(1R,3S,3aS,6aR)-3-(5-methyl-1-phenyl-1H-pyrazol-4-yl)-5-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(2-hydroxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-3-(1H-imidazol-2-yl)benzamide
N4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3S,4R)-1-[2-(5-acetylthiophen-3-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
5-{1-[4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
2-ethoxy-5-{2-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]pyrimidin-4-yl}benzoic acid
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
1-({5-[(5-ethylpyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
4-hydroxy-2-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]pyrimidine-5-carboxamide
4-fluoro-N-[(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]benzamide