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3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]urea
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1,9-dimethyl-4-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-methyl-1'-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
methyl 2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-6-(thiolan-3-yl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N,2,8-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]quinoline-4-carboxamide
ethyl 4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperazine-1-carboxylate
1-(3,3-diphenylpiperidin-1-yl)-2-hydroxyethan-1-one
N-[(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]-4-methoxybenzene-1-sulfonamide
4-[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-4-oxobutane-1-sulfonamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,3-benzothiazole-6-carboxamide
1-(2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)-1,4-diazepan-5-one
methyl (2S,4R)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[(phenylcarbamoyl)amino]pyrrolidine-2-carboxylate
1-(2,2-dimethylpropyl)-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyridin-2-yl}methanol
N-[2-methyl-2-(piperidin-1-yl)propyl]-5-propyl-1,3,4-oxadiazol-2-amine
N-[3-(1H-indol-1-yl)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
N-[(2S,4R,6S)-2-ethyl-6-(quinolin-4-yl)oxan-4-yl]benzamide
2-(1H-1,3-benzodiazol-1-yl)-N-(1-methyl-1H-indazol-3-yl)acetamide
(1R,5S)-6-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-carboxamide
5-(4-fluorophenyl)-2-methyl-4-{1-[4-(trifluoromethyl)benzoyl]piperidin-3-yl}pyrimidine
1-[(2,3-dimethoxyphenyl)methyl]-3-{[(2,2-dimethylpropyl)amino]methyl}-3-hydroxypiperidin-2-one
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(3-ethenylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-4-{1-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]ethyl}piperazine
(2R,6R)-4-[(2-cyclohexylpyrimidin-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-({1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
1-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-methoxy-2-phenylacetamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-benzyl-N3-ethyl-4-oxo-N5-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-cyclopropyl-N,N-bis(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(3S,4R)-1-(6-methyl-2-phenylpyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carbonitrile
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-3-ylmethyl)amine
2-(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N-{1-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
(2S,4S)-4-amino-N,N-diethyl-1-[(2-ethyl-1-benzofuran-3-yl)methyl]pyrrolidine-2-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
ethyl 4-[4-phenyl-1-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-imidazol-5-yl]-1H-pyrazole-3-carboxylate
3-[4-(3-phenylpropyl)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
4-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3-thiazol-2-amine
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[4-(methylamino)butyl]propanamide
N3-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
4-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]-N,N-dimethylpiperazine-1-carboxamide
3-(3-methoxypropyl)-3-(1-methylpiperidin-4-yl)-1-(1-phenylethyl)urea
2-{[(5-acetylpyridin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide