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1-cyclopropyl-N-(3-hydroxy-3-phenylpropyl)-N-methyl-1H-pyrrole-2-carboxamide
N-[(4-hydroxy-3-methoxyphenyl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-{[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
1,9-dimethyl-4-[3-(trifluoromethyl)pyridin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(methoxymethyl)-6-methyl-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,4-diazepane
4-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)morpholine
(2R,6S)-2,6-dimethyl-N-[3-(1H-pyrazol-5-yl)phenyl]morpholine-4-carboxamide
N-{3-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
3-(2-amino-1,3-thiazol-4-yl)-N-{2-[methyl(phenyl)amino]propyl}propanamide
2-[3-(pyridin-3-yl)azetidin-1-yl]-3-(pyrrolidine-1-carbonyl)pyridine
6-methyl-5-phenyl-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-ethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-6-oxopiperidine-3-carboxamide
(1S,5R)-6-(2,5-dimethylbenzoyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-(2,2-diethylmorpholin-4-yl)ethan-1-one
5-[1-(2-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-2-[2-(thiophen-2-yl)ethyl]piperidine-1-carboxamide
1-phenyl-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]cyclohexane-1-carboxamide
2-{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
5-({4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1H-indole
2-oxo-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
6-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
N-(cyclohexylmethyl)-4-oxo-1-(propan-2-yl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-2,4-dimethylpyrimidine
2-(3,4-dichlorophenyl)-4-(3-ethyl-1H-pyrazole-5-carbonyl)morpholine
1-(1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-3-phenylpropan-1-ol
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-1,3-dimethyl-1H-pyrazole-4-carboxamide
3-{[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
[4-methyl-5-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methanol
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N,N-diethyl-9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.5]undecane-3-carboxamide
2-[5-(3,4-dihydro-2H-1-benzopyran-3-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine
3-({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-(4-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-cyclopropyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-N-(1,3-thiazol-2-ylmethyl)acetamide
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
N-[(3S,4R)-4-(propan-2-yl)-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl]methanesulfonamide
1-({[1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
(2S,4R)-N-methyl-1-[(5-methylfuran-2-yl)methyl]-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(pyridin-3-yl)propanamide
N,N,4-trimethyl-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-cyclopropyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
7-(2-methoxyphenyl)-2-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(4-fluorophenyl)methyl]-2-methyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
(1R,5R)-6-(cyclobutylmethyl)-3-[4-(1H-imidazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane