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2-methyl-4-(1H-pyrazol-1-yl)-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
methyl 2-[(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)(methyl)amino]acetate
[(3R,4S)-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(3S,4S)-4-cyclopropyl-1-({[2-(4-methoxyphenyl)ethyl]carbamoyl}methyl)pyrrolidine-3-carboxylic acid
1-cyclopropanecarbonyl-4-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}piperidine
2-(dimethylamino)-2-(3-fluorophenyl)-N-(2-hydroxyethyl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
1-(2-methoxyethyl)-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1-methylcyclopropanecarbonyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(2S,4S)-4-amino-1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-N-methylpyrrolidine-2-carboxamide
6-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
(3R,5S)-1-benzyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-{3-[4-(1-phenyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}-2,3-dihydro-1H-imidazol-2-one
(2R,6R)-4-(2-ethoxyethyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(1S,5R)-6-(pyridin-2-ylmethyl)-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(hydroxymethyl)piperidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
4-(3-{[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
5-{3-[(3-chlorophenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}-1-methyl-1H-pyrrole-3-carbonitrile
(1S,5R)-3-(3-methoxypyrazin-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
1,9-dimethyl-4-[3-(thiophen-3-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-({4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}methyl)thiophene-2-carboxylic acid
2,5-dimethyl-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
N-benzyl-N-ethyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
N-cyclohexyl-4-[2-(piperazin-1-yl)acetamido]piperidine-1-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}propanamide
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
methyl 6-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]pyrazine-2-carboxylate
6-(methylamino)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
3-{[(2-aminopyridin-3-yl)methyl]sulfamoyl}-N-cyclopentylbenzamide
1-[2-(3-chlorophenyl)ethyl]-4-{[(1-ethyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-2-one
5-{[3-(4-fluorophenoxymethyl)piperidin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
2-methyl-3-({3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)quinoxaline
3-[2-(2,6-difluorophenyl)ethyl]-1-(ethanesulfonyl)piperidine
(2R,3R,6R)-5-{imidazo[1,2-b]pyridazine-3-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-(4-fluorophenyl)-2-methylpyrimidine
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-{[1-(dimethylsulfamoyl)-4-hydroxyazepan-4-yl]methyl}pyridine-4-carboxamide
(3S,4S)-4-cyclopropyl-1-[(5-propylfuran-2-yl)methyl]pyrrolidine-3-carboxylic acid
N-[(1-{[2-(methylsulfanyl)phenyl]carbamoyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]urea
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-(pyridin-4-yl)propanamide
2-(2-chloro-6-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-methyl-2-(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
2-{9-[(6-methylpyridin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
4-methyl-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-1,2,5-oxadiazole-3-carboxamide
6-{[(3R,4R)-4-hydroxypyrrolidin-3-yl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide