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4-(2-{1-[(6-chloropyridin-3-yl)methyl]piperidin-2-yl}ethyl)morpholine
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-6-methoxypyridine
N-(cyclopentylmethyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-benzyl-3-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
methyl 1-(3-{3-[(cyclopentylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
9-[5-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
dimethyl[3-(2-{1-[6-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)propyl]amine
1-[2-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)pyrimidin-4-yl]piperidin-3-ol
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](1H-indol-7-ylmethyl)methylamine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamide
1-(cyclopropylmethyl)-4-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperazine
1-({1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
4-benzyl-1-(3,5-dimethylbenzoyl)-3-ethyl-1,4-diazepan-5-one
3-(4-methyl-1H-pyrazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-3-carboxamide
(2R)-N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-amino-3-(ethylsulfanyl)propanamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}urea
N4-[(3-chlorophenyl)methyl]-N4-methyl-6-(4-methylpiperazin-1-yl)pyrimidine-2,4-diamine
1-(4-{2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
1-{[3-(2-methylphenyl)phenyl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
ethyl 1-(2,5-dimethylphenyl)-5-{[(1,2-oxazol-3-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
7-(4-chlorophenyl)-2-(4-hydroxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
3-cyclopropyl-1-[(4-methylphenyl)methyl]-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
1-[4-(difluoromethoxy)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-2-(trifluoromethyl)morpholine
8-[2-(morpholin-4-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-1H-pyrazole-5-carboxamide
N-[(8-methoxy-2H-chromen-3-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
1-(3-fluoro-4-methylbenzoyl)-3-(2-methoxyphenoxy)azetidine
(2S,5R)-1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethylpiperazine
1-[(2,3-dimethoxyphenyl)methyl]-3-{[(2-fluoroethyl)amino]methyl}-3-hydroxypiperidin-2-one
N-(2-methyl-1-benzofuran-7-yl)-4-[2-(morpholin-4-yl)ethyl]piperazine-1-carboxamide
1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-(hydroxymethyl)piperidin-3-ol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(4aS,7aR)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-methoxyethyl)-5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-1,2,4-oxadiazole
4-ethyl-3-{2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}piperazin-2-one
2-{4-[(4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenoxy}pyrimidine
2-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-hydroxyethyl)piperidine-2-carboxamide
4-methoxy-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-(2-aminopyrimidin-4-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
1-[4-({ethyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-{4-[1-(1,2,3-thiadiazole-4-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
3,7-dimethyl-11-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-3,7,11-triazaspiro[5.6]dodecane