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3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-(3-methylbutyl)piperidine
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
4-chloro-N-cyclopropyl-2-propanamido-N-(pyridin-2-ylmethyl)benzamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
5-[(1,3-benzothiazol-2-ylmethyl)amino]-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-(4-methylphenyl)-3-phenylpropan-1-one
N-butyl-N-[(5-methylthiophen-2-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
methyl 2-[4-(3-chlorophenyl)-3-oxopiperazine-1-carbonyl]piperidine-1-carboxylate
[(2,4-dimethoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
N-[3-(4-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
N,N,3-trimethyl-4-({[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}amino)benzamide
methyl 4-({4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)benzoate
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-(4-fluorophenyl)oxolan-3-yl]methyl})amine
6-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-9H-purin-2-amine
5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N-ethylpyrimidin-2-amine
4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2-(3-phenylpropyl)morpholine
8-(6-aminopyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 4-{1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carbonyl}piperazine-1-carboxylate
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(naphthalen-1-ylmethyl)-5-(1H-pyrazol-4-yl)-1,2,4-oxadiazole
3-(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-1-yl)phenol
6-(2-chlorophenyl)-2-(2-methylpiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(2S,4S)-4-amino-N-methyl-1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidine-2-carboxamide
(2S,4R)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidine
3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-pyrazol-5-amine
8-methoxy-2-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}quinoline
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
(3aS,6aR)-N-tert-butyl-2-oxo-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
N4,N4,5-trimethyl-N2-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrimidine-2,4-diamine
(3S)-N,N-dimethyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]azepan-3-amine
1-{3-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 4-{[(2-{1-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
2-[(cyclopropylmethyl)(propyl)amino]-N-(2-acetamidophenyl)acetamide
2-(2,2-diphenylethyl)-4-methanesulfonylmorpholine
8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-[2-(1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N,N-diethyl-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
N-[(3S,4R)-1-(5-acetylthiophene-2-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
(2S,4S,5R)-4-(dimethylcarbamoyl)-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
2-[2-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenoxy]ethan-1-ol
2-[2-({3-[(4-fluorophenyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
8-fluoro-3-[2-(1H-imidazol-4-ylmethyl)-3-oxopiperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
5-propyl-4-{4-[4-(pyridin-2-ylmethyl)piperazin-1-yl]piperidin-1-yl}pyrimidine
N-{4-methyl-2-[2-(propan-2-yloxy)acetamido]phenyl}cyclohexanecarboxamide
2-(1-{[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine