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N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-hydroxypropanamide
[(2S,6S)-4-[(6-methylpyridin-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
5-(4-acetylpiperazin-1-yl)-N-[(2-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-ethoxy-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
1-{2-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
(1R,5S,6R)-3-{[4-(1H-imidazol-1-yl)phenyl]methyl}-N-(pyridin-3-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-3-phenylbutanamide
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[1-(pyridin-2-yl)ethyl]amine
1-[4-(furan-2-yl)phenyl]-3-[3-(4-methylpiperazin-1-yl)propyl]urea
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(2S,4S)-4-amino-1-[2-(1H-1,3-benzodiazol-2-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
2-[4-(1-benzofuran-2-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
3-({[2-(4-hydroxyphenyl)ethyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-(2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}quinolin-6-yl)acetamide
N-(1-cycloheptylpiperidin-3-yl)-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
2-amino-1-(2-amino-4-{[(1-ethyl-1H-imidazol-5-yl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}acetamide
dimethyl({2-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-1-(5-methylfuran-2-yl)ethyl})amine
N,N-dimethyl-2-[3-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-5-yl]aniline
(3aR,6aR)-2-(furan-3-carbonyl)-5-(3-methylbut-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,9aR)-8-[(2,5-dimethylphenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(furan-2-ylmethyl)pyrrolidin-2-one
3-(3-chlorophenyl)-3-phenyl-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(benzyloxy)-8-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-4-(3-ethenylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-{3-[cyclohexyl(methyl)amino]propyl}-8-{spiro[2.3]hexane-1-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]pyrimidine
5-{2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-(3-methanesulfonamido-4-methoxyphenyl)urea
1-ethyl-N,2,5-trimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrrole-3-carboxamide
ethyl 3-{2-[(adamantan-1-yl)carbamoyl]acetamido}propanoate
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
2-({[(3R,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[2-(benzylsulfanyl)ethyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(thiophen-3-yl)acetamide
N-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
N-(2,2-dimethyloxan-4-yl)-1-{4-[(dimethylsulfamoyl)amino]phenyl}piperidin-4-amine
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
1-[2-(dimethylamino)ethyl]-N-[2-(4-methylphenyl)propan-2-yl]-6-oxopiperidine-3-carboxamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
1-[4-(furan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(4H-1,2,4-triazol-4-yl)propanamide
2-(2-hydroxyethyl)-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[(3-hydroxypiperidin-1-yl)methyl]-N-[(1-phenylcyclohexyl)methyl]-1,2-oxazole-3-carboxamide
N,N-dimethyl-1-(2-methylpropyl)-5-{[(3,4,5-trifluorophenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{4-[2-(4-methylpentyl)morpholin-4-yl]pyridin-2-yl}methanol