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5-methyl-1'-[4-(pyrrolidin-1-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(2R,3R,6R)-5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-1,2-dihydroisoquinolin-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(4-fluoro-2-methylphenyl)-3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)propanamide
[(1,2-dimethyl-1H-imidazol-5-yl)methyl](methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
2-[benzyl(methyl)amino]-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1,2-dihydroquinoxalin-2-one
3-{1-[2-(azepan-1-yl)acetyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
5-ethyl-1'-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{3-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
2-ethoxy-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)benzamide
(4aR,7aS)-4-(2-methoxypyridine-4-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-{1-[3-(2-methoxyethoxy)phenyl]-1H-imidazol-2-yl}phenol
(4aR,7aS)-1-benzyl-4-(dimethyl-1,3-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 5-[2-amino-3-cyano-6-(1-methyl-1H-pyrrol-3-yl)pyridin-4-yl]-2-hydroxybenzoate
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-oxo-2-phenylacetamide
2-[5-(5-methoxyfuran-2-yl)-3-methyl-1H-1,2,4-triazol-1-yl]pyridine
3-(3-fluorophenyl)-4-(8-fluoroquinoline-2-carbonyl)piperazin-2-one
N-{2-methoxy-4-[3-(1H-pyrazol-1-yl)phenyl]phenyl}acetamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]quinoline-3-carboxamide
(3R,4S)-1-(6-chloro-2H-chromene-3-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
N-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}methyl)pyridine-4-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}morpholine
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]propanoate
3-cyclohexyl-N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1H-pyrazole-4-carboxamide
6-[(diethylamino)methyl]-N-[1-(4-hydroxyphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-benzyl-2-(2-ethylpyrimidin-5-yl)-N-methylquinoline-4-carboxamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(1H-indazol-1-yl)acetamide
5-acetyl-2,4-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-pyrrole-3-carboxamide
1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
3-({1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidin-4-yl}oxy)pyridine
9-[(5-ethylpyridin-2-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}thiophene-2-carboxylic acid
N-butyl-N-(furan-2-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
7-[(3-methylphenyl)methyl]-2-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
4-(2H-1,3-benzodioxole-5-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
[(5-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
6-fluoro-2-oxo-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-{[2-(4-cyano-4-phenylpiperidine-1-carbonyl)phenyl]amino}acetic acid
1-[(3-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-benzyl-N-methyl-1H-pyrazole-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2,4-dimethylphenoxy)-3-{[1-(1-methylcyclopropyl)propan-2-yl]amino}propan-2-ol