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N-{4-[4-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}benzenesulfonamide
N-benzyl-N,1-dimethyl-5-[methyl(thiophen-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-ethylpiperidine
N,N,4-trimethyl-3-({[2-(4H-1,2,4-triazol-4-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(2,5-dimethylphenoxy)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]propanamide
5-oxo-1-[4-(1H-pyrazol-5-yl)phenyl]pyrrolidine-3-carboxylic acid
3-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}benzoic acid
4-{3-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-methyl-1,2-dihydrophthalazin-1-one
N-methyl-4-(1H-pyrazol-3-yl)-N-(quinolin-5-ylmethyl)benzamide
1-{3-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-4-(morpholin-4-yl)phenyl}ethan-1-one
4-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-2,6-dimethoxyphenol
(2S,4S)-4-amino-N-ethyl-1-(1H-indole-3-carbonyl)pyrrolidine-2-carboxamide
2,6-dimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-4-carboxamide
N-[(1-phenylcyclopentyl)methyl]-9H-purin-6-amine
(3R,4S)-4-cyclopropyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-amine
2-(4-{2-[(2-methoxyphenyl)methoxy]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenylacetamide
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]thieno[2,3-d]pyrimidine
N-[(5-ethylpyridin-2-yl)methyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
1-(4-methyl-1H-pyrrole-2-carbonyl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-[3-chloro-5-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
5-chloro-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(2-ethylphenoxy)-N-{2-[2-(methylcarbamoyl)ethyl]phenyl}azetidine-1-carboxamide
5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
3-[3-(1H-imidazol-1-yl)propyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-cyclohexylethyl)-3-hydroxy-3-[(4-methoxypiperidin-1-yl)methyl]piperidin-2-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-(2-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}phenyl)ethan-1-one
ethyl 1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
1-(1-benzofuran-2-ylmethyl)-3-(3,4-dimethoxybenzoyl)piperidine
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-3-(2-ethyl-1H-imidazol-1-yl)propanamide
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
3-[2-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)ethyl]pyridine
4-(5-methylpyridin-2-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-ol
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}azocane
8-methoxy-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-(3-phenyl-1H-pyrazole-5-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
N-[(2-aminopyridin-3-yl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
5-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
N,N,4-trimethyl-5-(4-phenylpiperidine-1-carbonyl)pyrimidin-2-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(6-methylpyridazin-3-yl)piperazin-2-yl}ethan-1-ol
5-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}-2,1,3-benzothiadiazole
(3R)-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
7-(3,6-dimethylpyrazin-2-yl)-4-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]ethan-1-one