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2-amino-N-(1-benzothiophen-2-ylmethyl)-3-ethyl-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(4aS,8aR)-6-(ethanesulfonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
3-(2-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
N-[(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-4-yl)methyl]acetamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
methyl 2-(3-{[(4-methoxyphenyl)methyl]carbamoyl}-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl)acetate
2-amino-4-(3-hydroxy-4-methoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-(3-ethoxypropyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,9S)-11-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-(2-{1-[2-(1H-1,3-benzodiazol-2-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-6-(methoxymethyl)pyridine-2-carboxamide
2-{4-[3-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
(2S,4R)-4-cyclopropaneamido-N,N-diethyl-1-(4-fluorobenzoyl)pyrrolidine-2-carboxamide
2-methoxy-1-{4-[(2-methyl-1H-imidazol-4-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
[3-(2-phenoxyethyl)-1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]methanol
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
methyl (2S,4R)-4-[(phenylcarbamoyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
N-[3-(dimethylamino)propyl]-1-(5-fluoro-2-methylbenzenesulfonyl)-N-methylpiperidin-3-amine
2-(2-{[1-(pyrimidin-2-yl)piperidin-4-yl]amino}ethyl)-3,4-dihydroquinazolin-4-one
8-(5-acetylpyridin-2-yl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-(piperidin-4-ylmethyl)cycloheptanamine
N-(3-hydroxypropyl)-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
({[2-(2-fluorophenoxy)pyridin-3-yl]methyl}sulfamoyl)dimethylamine
N-[(2-aminopyridin-3-yl)methyl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-(cyclopropylmethyl)-5-(3-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-methanesulfonyl-3-[2-(4-methoxyphenyl)ethyl]piperidine
3-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}-N-(pyridin-3-yl)propanamide
2-oxo-N-(2,2,6-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1,2-dihydroquinoline-4-carboxamide
2-chloro-5-acetamido-N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
propan-2-yl 4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-[(3-methoxyphenyl)methyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-4-(piperidin-1-yl)benzamide
(1S,5R)-3-(3-chlorobenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-ethyl-5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-1,3-thiazol-2-amine
(1S,5R)-3-methyl-6-(3,5,7-trimethyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[2-oxo-2-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)ethyl]-1,3-thiazolidine-2,4-dione
6-methyl-5-{5-[1-(propan-2-yl)azetidin-3-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(3-methoxyphenyl)piperidine
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(dimethylamino)ethyl]-N-methyl-3-phenylpropanamide
5-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]pyrrolidin-2-yl}-N,N-dimethylthiophene-2-carboxamide
1-(methoxymethyl)-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]cyclobutane-1-carboxamide
1-acetyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)piperidine-3-carboxamide
N-benzyl-N-methyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
N-[3-(3-fluorophenyl)phenyl]-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(1S,5R)-6-(3-methoxy-2-methylbenzoyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}benzamide
3-ethoxy-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazine