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6-[1-(2,6-dimethylquinoline-4-carbonyl)piperidin-3-yl]pyrimidin-4-ol
(3R)-1-({1-[1-(3-methylquinolin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-4-hydroxy-1-methylpiperidine-4-carboxamide
2-(5-{4-[1-(dimethylamino)ethyl]phenyl}-4-phenyl-1H-imidazol-1-yl)-2-methylpropane-1,3-diol
(1S,5R)-3-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-fluoro-N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
1-methyl-2-(2-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)-1H-1,3-benzodiazole
3-(1-methylpiperidin-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-({4-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}(methyl)amino)ethan-1-ol
2-amino-6-(1,2-dimethyl-1H-indol-3-yl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
ethyl 1-(5-methoxy-5-oxopentanoyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
[(3R,4R)-1-(2-chloro-5-fluorobenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-{4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[(2-fluorophenyl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
{1-[(4-fluorophenyl)methyl]-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl}(phenyl)methanol
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-[1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
3-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
4-methoxy-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}benzene-1-sulfonamide
({5-[1-(3-ethoxybenzoyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[4-(ethylsulfanyl)phenyl]-4-[1-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
2-(4-methyl-1H-imidazol-5-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazole
3-cyclohexyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
4-methyl-5-[3-(2-methylphenyl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
methyl 5-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-[3-(2-ethylphenoxy)azetidin-1-yl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
1-(4-tert-butylbenzoyl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
(3S,4R)-4-(2-methylphenyl)-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-3-carboxylic acid
N-benzyl-N-methyl{[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]amino}sulfonamide
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-fluorobenzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(3-phenylpropyl)acetamide
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
4-ethyl-1-methyl-3-[1-(2-methyl-2-phenylpropanoyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
{4-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]phenyl}methanol
N-[4-(4-{[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-benzyl-4-(1-ethyl-1H-imidazol-2-yl)piperidine
(1S,5R)-3-(2-fluorobenzenesulfonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopentyl-4-oxo-4-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}butanamide
2-(2-methoxy-4-methylphenoxymethyl)-4-(2-phenylazetidine-1-carbonyl)-1,3-oxazole
N-(3,4-dimethylphenyl)-1-(quinoxaline-6-carbonyl)piperidin-3-amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-fluoro-5-sulfamoylbenzamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(4-methylphenyl)propan-1-one
2-[2-(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-3-(pyridin-3-yl)propan-1-one
(1S,5R)-3-[(3-chlorophenyl)methyl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide