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3-(4-methoxyphenyl)-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
ethyl 3-benzyl-1-{[2-(trifluoromethyl)phenyl]carbamoyl}piperidine-3-carboxylate
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(morpholin-4-yl)butan-1-one
(2S,4S)-4-amino-N-ethyl-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrrolidine-2-carboxamide
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one
2-methoxy-5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[(thiolan-3-yl)amino]pyridine-3-carboxamide
N-{2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]propan-1-ol
N-[cyclohexyl(thiophen-2-yl)methyl]-1-cyclopropanecarbonylpiperidine-4-carboxamide
N5-cyclohexyl-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(thiophene-3-carbonyl)-1,4-diazepan-2-one
(1R,6S)-9-methyl-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-methyl-3-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}-1H-1,2,4-triazole
N2-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
3-(5-{[3-(5-methylfuran-2-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
2-methoxy-4-({[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amino)pyridine-3-carbonitrile
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(propan-2-yloxy)propan-1-one
2-(3-hydroxyphenyl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
1-cyclobutanecarbonyl-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylic acid
3-(2-hydroxyphenyl)-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(2-hydroxyethyl)-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
5-fluoro-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(morpholin-4-yl)pyrimidin-2-amine
4-({[(6-chloropyridin-3-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-pyrazol-4-yl)benzamide
(2S)-2-(2,3-difluorophenyl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}acetic acid
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-[4-(1,4-dithiepan-6-yl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(2-acetamidoethyl)-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
8-[2-(propan-2-yloxy)acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[3-(1-phenylcyclopropyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-[(3S,4R)-1-(3-hydroxy-4-methylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(2R,6S)-4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]-2,6-dimethylmorpholine
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[3-(pyridin-3-yloxy)propyl]benzamide
3-(4-chlorobenzoyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine
(2R,3R,6R)-3-(4-fluorophenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
6-methyl-8-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(2,5-dioxoimidazolidin-4-yl)acetamide
methyl 2-[8-(butan-2-yl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-[3-(methylsulfanyl)propyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(pyrrolidin-1-yl)pentan-1-one
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide