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({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)(pyrimidin-2-ylmethyl)amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-ethyl-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
2-methyl-9-(oxane-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-(3,5-dimethylphenyl)-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-cyclopentyl-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(2S)-2-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanamide
4-[(3-chlorophenyl)methyl]-7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{2-methylthieno[3,2-d]pyrimidin-4-yl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
4-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4-[4-(4-ethylpiperazine-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
1-{3-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
4-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-6-(1H-pyrazol-1-yl)pyrimidine
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
1-[1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]pyrrolidin-2-one
(butan-2-yl)[(5-ethylpyridin-2-yl)methyl](thiophen-3-ylmethyl)amine
2-cyclopropyl-5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-3,4-dihydropyrimidin-4-one
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[1-(phenoxymethyl)cyclopropyl]methyl}acetamide
3-methoxy-N-[2-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
2-[(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)methyl]-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[1-(2-chlorophenyl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N,5-dimethyl-7-(trifluoromethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-(3-{2-amino-3-cyano-7-methyl-5H,7H-thieno[3,4-b]pyridin-4-yl}phenoxy)acetamide
4-(furan-2-ylmethyl)-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-oxo-4H-chromene-2-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(4-fluoro-3-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N,N-dimethyl-3-{[(3-phenyl-1H-pyrazol-5-yl)methyl]sulfamoyl}benzamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(thian-4-yl)benzamide
N-[(1-benzylpiperidin-4-yl)methyl]-2-(3-hydroxypiperidin-1-yl)-N-methylacetamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-(oxolan-3-yl)-5-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-1,2,4-oxadiazole
3-{ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfamoyl}-N-[2-(methylamino)ethyl]benzamide
1-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-[4-(1H-imidazol-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methoxybenzamide
6,8-dimethyl-2-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
(3R,4R)-4-[(6-chloroquinolin-2-yl)amino]piperidin-3-ol
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
[(5-cyclopentylthiophen-2-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-[4-(dimethylamino)azepan-1-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-(2,3-difluorophenoxymethyl)-N-ethyl-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
7-fluoro-3-methyl-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1-benzofuran-2-carboxamide
2-methyl-7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N,2,8-trimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}quinoline-4-carboxamide
2-(2,4-difluorophenoxy)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
8-(6-aminopyrimidin-4-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-chloro-3-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one