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2-methyl-4-phenyl-9-(pyridazine-3-carbonyl)-2,9-diazaspiro[5.5]undecane
N-[(2-chlorophenyl)methyl]-2-(2-oxoazepan-1-yl)-N-(prop-2-en-1-yl)acetamide
2-ethyl-N-methyl-N-[3-(oxolan-2-yl)propyl]pyrimidine-5-carboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-4-(4-methylphenyl)piperazine-1-carboxamide
N-ethyl-2-{4-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]phenyl}acetamide
5-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
(2S)-2-({4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}formamido)-4-methylpentanamide
4-cyano-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
ethyl 4-[5-(3-acetylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
7-methyl-2-(4-phenylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1-(propan-2-yl)-1H-pyrrole-2-carboxamide
4-chloro-N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-1-methyl-1H-pyrazole-3-carboxamide
4-[3-(4,5-diphenyl-1H-imidazol-1-yl)propanoyl]piperazin-2-one
4-(4-chlorophenyl)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-ol
N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
2-methyl-4-propyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
2-{cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-N-[1-(4-methylphenyl)ethyl]acetamide
4-(2-{[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}ethyl)benzoic acid
4-(4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
(2S)-2-amino-1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]hexan-1-one
ethyl 3-[(2-methylphenyl)methyl]-1-(pyridine-3-carbonyl)piperidine-3-carboxylate
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(1,4-dioxan-2-ylmethyl)[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]methylamine
N,N-dimethyl-5-{1-[1-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(furan-3-ylmethyl)methylamine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[3-(methylsulfanyl)propyl]propanamide
5-(4-tert-butylbenzoyl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl 4-({[(1-ethylpyrrolidin-2-yl)methyl]carbamoyl}amino)-3-methylbenzoate
2-[(1S,5R)-3-(2,4-dimethylpyrimidine-5-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
6-{3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}-N-[(2-fluorophenyl)methyl]acetamide
N-[3-(4-cyclopentyl-1,4-diazepan-1-yl)-3-oxopropyl]-2-fluorobenzamide
N-[2-(benzylsulfanyl)ethyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
(3aS,7aR)-2-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-[1-(3-hydroxyadamantan-1-yl)ethyl]-1H-imidazole-2-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(3S,4S)-4-cyclopropyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyrrolidine-3-carboxylic acid
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-5-methyl-1,3-oxazole-4-carboxamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-(2-hydroxypropyl)-N-methyl-1,2-oxazole-3-carboxamide
4-[4-(2-cyclopentylacetyl)piperazin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(methylamino)acetamide
3-[(tert-butylamino)methyl]-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
N,3,5,7-tetramethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-indole-2-carboxamide