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4-[3-fluoro-2-(morpholin-4-yl)pyridin-4-yl]phenol
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidine
N-(3-chloro-4-methoxyphenyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
8-(1-benzofuran-5-ylmethyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(1S,2R)-2-[(1-benzoylpiperidin-4-yl)amino]cyclobutyl]-3-ethyl-1H-pyrazole-4-carboxamide
(2S)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(methylamino)propan-1-one
N4-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-cyclopentyl-6-oxo-N-[3-(4H-1,2,4-triazol-4-yl)propyl]piperidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-methylthiophene-2-carboxamide
5-[2-(2,3-dimethylphenoxy)ethyl]pyridine-3-carboxamide
3-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3S,4S)-4-(piperidin-1-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-hydroxy-4H-pyran-4-one
(3S,4S)-1-[2-(methylsulfanyl)benzoyl]-4-propylpyrrolidine-3-carboxylic acid
N-[(3R,5S)-5-(2,5-dihydro-1H-pyrrole-1-carbonyl)pyrrolidin-3-yl]-3,5-dimethoxybenzamide
[(dimethyl-1,2-oxazol-4-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
(3S,4S)-1-(furan-2-ylmethyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
3-acetamido-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}benzamide
N-benzyl-3-chloro-N-ethyl-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
N2,N2-dimethyl-N5-(1-phenylpiperidin-4-yl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
[(4-fluorophenyl)methyl][(3-methyl-1H-pyrazol-5-yl)methyl](pyridin-4-ylmethyl)amine
2-(4-{[2-(2,4-difluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenoxy)ethan-1-ol
3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
4-(2,6-dimethylpyrimidine-4-carbonyl)-1-(2-methylphenyl)piperazin-2-one
2-amino-4-(4-hydroxy-2-methoxyphenyl)-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
6-(2-methoxyphenyl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyridazin-3-amine
4-{[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}-1-ethylpiperazin-2-one
3-{1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}-4H-chromen-4-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
N-({5-[(5-phenylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
(2R,6R)-4-[3-(dimethylamino)-2,2-dimethylpropyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-methyl-4-({1-phenyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}methyl)piperidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-acetamido-N,3-dimethylbenzamide
(1-benzothiophen-2-ylmethyl)(methyl){[4-({1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
3-methoxy-2-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}phenol
2-[2-(2-methoxyquinolin-3-yl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(5-propyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
8-[6-(morpholine-4-carbonyl)pyrazin-2-yl]quinoline
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)benzamide
(1-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
2-methoxy-3-{3-[(1-methylpiperidin-4-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}pyridine
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-[5-(2-methylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]pentanoic acid