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3-(2,5-dioxoimidazolidin-4-yl)-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]propanamide
3-{5-[2-(1H-pyrazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridazine
4-{[(2R,5S)-5-[(3-ethoxyphenyl)methyl]oxolan-2-yl]methyl}morpholine
ethyl 1-[2-(2H-1,3-benzodioxol-5-yl)acetamido]piperidine-3-carboxylate
1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-(furan-2-ylmethyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-3-carboxamide
N-ethyl-N-methyl-5-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-{4-phenyl-1-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-imidazol-5-yl}pyrimidin-2-amine
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
6-{2-[(dimethylamino)methyl]phenyl}-N-(propan-2-yl)pyridazin-3-amine
(2E)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-(furan-2-yl)prop-2-enamide
N-(1,3-benzothiazol-5-yl)-3-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
(2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-8-methylquinolin-3-yl)methanol
6-(benzyloxy)-4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
4-({ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-2,6-dimethylphenyl acetate
N-[(3R,5S)-1-cyclobutanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-imidazole-5-carboxamide
4-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,2,3-thiadiazole-5-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(6-methylpyridine-2-carbonyl)piperidine-3-carboxylate
1-(2-methoxyphenyl)-2,2-dimethyl-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
6-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-(1H-indol-4-ylmethyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
N4-[(2-methyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[4-(1H-indol-2-yl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
3-fluoro-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2,6,8-trimethyl-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]quinoline
5-[1-(4-acetamido-3-methoxyphenyl)-1H-imidazol-2-yl]thiophene-2-carboxylic acid
(1r,4r)-4-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)cyclohexan-1-ol
N,N-diethyl-1-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-methyl-3-(quinolin-6-yl)benzamide
N,3,4,7-tetramethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-indole-2-carboxamide
2-(dimethylamino)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-fluorophenyl)acetamide
3-[8-(1,1-dioxo-1λ6-thiane-4-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
methyl (2S)-2-cyclopropyl-2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}acetate
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-ethylpyrimidin-2-amine
5-(cyclohexylamino)-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 1-ethyl-5-(2-oxo-2-phenylacetyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3aR,6aR)-2-(2-methoxyethyl)-5-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
3-[(3-chlorophenyl)methyl]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
2-(1-benzofuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-(azepane-1-carbonyl)-1-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methanesulfonyl-N-[2-(2-phenoxyethoxy)phenyl]acetamide
N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-[3-(2-methylpropyl)-1-phenyl-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
6-methyl-1-[(3-methylpyridin-4-yl)methyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}pyridine
3-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}-1-[4-(pyridin-3-yloxy)phenyl]urea
[1-(4-chloro-2-methoxybenzoyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol