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methyl 5-{7-[(3-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-5-oxopentanoate
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-1-(morpholin-4-yl)ethan-1-one
(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)(pyridin-3-ylmethyl)amine
1-(2,6-dimethylpyridin-4-yl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazine
2-{3-[3-(5-acetylthiophen-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-{4-[(4-methyl-3-phenylpiperazin-1-yl)methyl]phenyl}acetamide
(4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}morpholin-2-yl)methanamine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-benzyl-5-hydroxy-N-methyl-1-oxa-9-azaspiro[5.5]undecane-9-sulfonamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-({[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}methyl)-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
1-[2-({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}amino)ethyl]piperidin-4-ol
1-(4-methylphenyl)-4-[2-(propan-2-yloxy)propanoyl]piperazin-2-one
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-[2-(3-fluorophenyl)ethyl]piperidine
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
6-(4-methylpiperazin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
2-{[(2-methylphenyl)methyl]sulfanyl}-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
N-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methylpyrrolidine-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(pyridin-3-yloxy)ethyl]benzamide
4-methyl-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(propan-2-yl)-5-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
7-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2,2,2-trifluoro-N-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylformamido}ethyl)acetamide
2-(2,4-difluorophenoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
3-[(3-hydroxypiperidin-1-yl)methyl]-N-(6-methoxypyridin-3-yl)benzamide
1-methyl-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1H-1,2,3-benzotriazole
6-methyl-5-[5-(5-methyl-2-phenylfuran-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-{1-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1H-imidazol-2-yl}benzonitrile
3-(3,4-difluorophenyl)-5-(thiolan-3-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
9-[3-(4-ethylphenyl)propanoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3,5-dimethoxyphenyl)-2-hydroxyethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
{4-[(3-methoxyphenyl)methyl]-1-[(E)-2-phenylethenesulfonyl]piperidin-4-yl}methanol
8-(2,2-dimethylbutanoyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-[(1R,5R)-6-[(2-ethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-4-carboxamide
(1S,5R)-3-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(5-ethylfuran-2-yl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[2-(benzenesulfonyl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-[4-(1H-pyrazol-3-yl)benzoyl]-4-(1,3-thiazol-2-yl)piperazine
4-{4-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]phenyl}-2-methylbut-3-yn-2-ol
4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-3,5-dimethyl-1,2-oxazole
3-methyl-7-[3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
1-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-3-(4-methoxy-2-methylphenyl)-1-methylurea
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(methylsulfanyl)ethyl]acetamide