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5-(2,6-difluorophenoxymethyl)-N-[(3,4-difluorophenyl)methyl]-1,2-oxazole-3-carboxamide
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-methylpyridine-3-carboxylic acid
6-ethoxy-3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}-1,2-dihydroquinolin-2-one
3-{2-[2-(2-methoxypyrimidin-5-yl)-1H-imidazol-1-yl]ethyl}-1H-indole
(4aS,7aR)-1-(4-methoxy-3-methylbenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-4-(3-fluorophenyl)-1-(2-methoxypyridine-4-carbonyl)pyrrolidine-3-carboxylic acid
5-ethanesulfonamido-N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
4-fluoro-3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
1-cyclopentyl-5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
1-(1H-indole-5-carbonyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
4-[(2-ethylpyrimidin-4-yl)methyl]-2-(pyridin-3-yl)morpholine
3-{5-[2-(carbamoylamino)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-cyclopentylpropanamide
5-(4-chlorophenyl)-4-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-pyrazole-3-carboxamide
2-(3-ethyl-1H-pyrazol-5-yl)-1-[(4-phenyloxan-4-yl)methyl]-1H-imidazole
1-(2,5-dimethylpyrimidin-4-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-methyl-8-(3-phenyl-1,2-oxazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(4-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
3-cyclopropyl-1-(3-fluorophenyl)-5-(methoxymethyl)-1H-1,2,4-triazole
6-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-(methoxymethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}cyclobutane-1-carboxamide
3-{[ethyl(methyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-phenylpropanamide
5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-2-[4-(trifluoromethyl)phenyl]-1,3-oxazole
2-[5-(1-ethylpiperidin-3-yl)-4-phenyl-1H-imidazol-1-yl]acetamide
1-(3-aminoazepan-1-yl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
(1S,4S)-5-(1-benzylpiperidin-4-yl)-2-(5-chloro-2-methoxyphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(3-methoxyphenyl)-1-[2-(methylsulfanyl)benzoyl]pyrrolidine
(4aS,8aS)-2-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-decahydroisoquinolin-4a-ol
N3-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-1,3-dicarboxamide
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propanamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(propan-2-yloxy)ethan-1-one
4-(2-cyanophenyl)-N-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)piperazine-1-carboxamide
2-[2-(methylsulfanyl)acetyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-methoxypyrimidin-2-yl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(carbamoylmethyl)-N-[(1R,2S)-2-phenylcyclohexyl]piperidine-4-carboxamide
1-[2-(4-chlorophenyl)ethyl]-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]piperidin-2-one
3-(2-fluorophenyl)-1-methyl-3-{2-oxo-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
3-[1-(adamantan-1-yl)piperidin-4-yl]-N-phenylpropanamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-3-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxy-2-methylpropan-1-one
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-hydroxyethan-1-one
2-[(ethylsulfanyl)methyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3R,4R)-4-[4-(2-phenylethyl)piperazin-1-yl]-1-(3,3,5,5-tetramethylcyclohexyl)piperidin-3-ol
(3aS,6aS)-2-ethyl-5-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(oxolan-2-ylmethyl)-N-propyl-4-(1H-pyrrol-1-yl)benzamide
N-[4-(4-{[(6-methylpyridin-2-yl)methyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
3-cyclopentyl-1-({1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)urea
2-ethoxy-4-[1-(pentan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenol