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3-{3-[3-(thiophen-2-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrrole-3-carboxamide
4-(3-methoxypiperidine-1-carbonyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine
3-(2-ethyl-6-methylphenyl)-1-methyl-1-(oxan-2-ylmethyl)urea
2-amino-8-hydroxy-4-(2-methoxypyrimidin-5-yl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-cyclopropyl-3-(1-phenyl-1H-pyrazol-5-yl)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-3-(2-oxopyrrolidin-1-yl)benzamide
(1R,5S,6R)-3-cyclopentyl-N-[(3-methylphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}(methyl)amino)propane-1,2-diol
(3S)-3-benzyl-4-[3-(methylsulfanyl)propyl]piperazin-2-one
2-amino-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,3-benzothiazole-5-carboxamide
2-(4-tert-butylphenoxymethyl)-4-hydroxy-N-(oxolan-3-ylmethyl)pyrimidine-5-carboxamide
[(2S,6S)-4-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
5-ethyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-amino-4-(5-tert-butyl-1H-pyrazol-3-yl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
4-(4-phenyl-1H-imidazol-5-yl)benzamide
4-{[3-(cyclopentylcarbamoyl)propanamido]methyl}benzoic acid
N-benzyl-6-[4-(cyclopropylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}(3-phenylpropyl)(pyridin-4-ylmethyl)amine
5-tert-butyl-4-({1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}methyl)furan-2-carboxamide
(3-{[1-(quinoline-6-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
4-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-1,2,2-trimethylpiperazine
1-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-2-phenylethan-1-one
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
N-[4-(5-ethylfuran-2-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]methanesulfonamide
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4-methyl-1,3-thiazol-2-amine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(4aR,7aS)-4-[(2,4-difluorophenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-acetyl-8-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{4-[4-(ethanesulfonyl)piperazin-1-yl]-6-ethylpyrimidin-2-yl}morpholine
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
3-[2-amino-4-methyl-6-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)pyrimidin-5-yl]propanoic acid
2-[2-(diethylamino)acetyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-{[4-(3-chlorophenyl)-5-{[methyl(quinolin-4-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
2-benzyl-N-methyl-N-(quinolin-4-ylmethyl)-1,3-thiazole-4-carboxamide
2-[1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
6-chloro-N,N-dimethyl-3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[1-(5-chloro-2-methoxyphenyl)-5-(morpholin-4-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
[(6-methoxypyridin-3-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
3-[methyl(1-methylpyrrolidin-3-yl)amino]-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
2-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)-2-(oxan-4-yl)acetamide
2-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
2-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one