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4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(2-chlorophenyl)-3-cyclopropyl-5-(methoxymethyl)-1H-1,2,4-triazole
4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]thiomorpholine
6-methyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-(1,3-dimethyl-1H-pyrazol-4-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(1H-imidazol-1-yl)-1-[2-(3-methylphenoxy)acetyl]piperidine-4-carboxylic acid
2-cyclopropyl-9-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[2-(cyclopentyloxy)phenyl]methyl}-1-methylpiperazin-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidin-2-amine
ethyl 1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine-3-carboxylate
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(4-methoxypyrimidin-2-yl)piperazin-2-yl}ethan-1-ol
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[(methylsulfanyl)methyl]piperidine
N-methyl-5-propyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
(4S)-4-(methoxymethyl)-1-[3-(2-methoxyphenoxy)propyl]-3,3-dimethylpiperidin-4-ol
5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
3-chloro-N,6-dimethyl-N-[2-(morpholin-4-yl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(4-ethoxy-2-fluorophenyl)-3-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]urea
3-(1H-imidazol-2-yl)-N-(1,2-oxazol-3-ylmethyl)benzamide
3-fluoro-N-(isoquinolin-5-ylmethyl)-N-methylpyridin-4-amine
3-tert-butyl-1-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)urea
N,2,5-trimethyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1,3-thiazole-4-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methylazepane-2-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2,2-diphenylethan-1-one
1-[2-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
1-cyclopropanecarbonyl-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
N-methyl-3-(morpholin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
6-(azepan-1-yl)-N-(1,4-dioxan-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
8-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-dimethyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methoxyphenol
N-(3-{2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)acetamide
(3R,4R)-4-cyclobutyl-3-methyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-ol
1-cyclopentanecarbonyl-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
N-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
2-(2-chlorophenoxy)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
2-(5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
methyl 5-[4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-5-oxopentanoate
[1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
4-({8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
[1-(3-methoxypyrazin-2-yl)-4-(2-phenylethyl)piperidin-4-yl]methanol
3-hydroxy-1-(2-phenylethyl)-3-{[(thiophen-3-ylmethyl)amino]methyl}piperidin-2-one
2-{imidazo[1,2-a]pyridin-3-ylmethyl}-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-ethyl-8-[2-(morpholin-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
4-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one