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2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]acetamide
8-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1-(propan-2-yl)-1H-pyrazole
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-3-ol
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[1-(2-methoxyphenyl)-1H-imidazol-2-yl]benzonitrile
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-4-(1H-pyrazol-4-yl)butanamide
2-[({1-[(2,3-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)(methyl)amino]-N-methylacetamide
3-hydroxy-3-({[(2-methoxyphenyl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-[2-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)ethan-1-one
[3-(2-methoxyethyl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]methanol
4-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methyl-1,3-oxazole
9-{[3-(trifluoromethyl)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
3-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]-2,8-diazaspiro[4.5]decane
3-cyclopropyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-[4-(2,4-dimethylpyrimidine-5-carbonyl)piperazin-1-yl]-4-phenylpyrimidine
methyl 2-{[7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]sulfonyl}benzoate
N-(3-phenylprop-2-yn-1-yl)-N-propyl-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
(1R,5S,8S)-3-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
5-{[benzyl(methyl)amino]methyl}-N-cyclopropyl-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidine-3-carboxylate
4-(1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-methyl-1,4-diazepane
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
5-[4-(ethylsulfanyl)phenyl]pyrimidin-2-amine
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
(4aR,7aS)-1-acetyl-4-[(2-fluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,2-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]benzamide
2-[4-(2-aminopyrimidin-4-yl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-[2-(2-phenyl-1,3-thiazol-5-yl)-1H-imidazol-1-yl]acetamide
4-methyl-3-({2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]acetamido}methyl)benzoic acid
methyl 2-({3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-8-carbonyl}amino)acetate
5-[5-(2-chloro-5-fluorophenyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(4-fluoropiperidine-1-carbonyl)-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2S)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]methanol
2-(2-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-hydroxy-4-methoxybenzamide
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}piperidin-4-ol
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
N-tert-butyl-3-(3-chlorobenzoyl)piperidine-1-carboxamide
1-[2-(3-methoxypropyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3,5-dimethoxy-2-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}benzoic acid
[(3R,4R)-1-(5-fluoro-2-methoxybenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(2-phenylethyl)-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
3-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(quinolin-3-ylmethyl)acetamide