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2-(4-ethylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
1-{3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}ethan-1-ol
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-(2-{[1-(carbamoylmethyl)piperidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
1-(2-methoxyethyl)-1-[(3-methoxyphenyl)methyl]-3-(2-methyl-1H-1,3-benzodiazol-6-yl)urea
N-(furan-2-ylmethyl)-5-{[(4-methoxyphenyl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 6-(3-chloro-4-fluorobenzoyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl[(1-methyl-1H-indol-2-yl)methyl][1-(pyridin-2-yl)ethyl]amine
1-(5-fluoro-2-methoxyphenyl)-3-{[1-(methoxymethyl)cyclopentyl]methyl}urea
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2,1-benzoxazole-3-carboxamide
7-(2-methoxyphenyl)-2-[(2-methylpropanesulfonyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[4-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)phenyl]ethan-1-amine
methyl 2-{[(3,4-difluorophenyl)methyl]sulfamoyl}-6-(pent-4-enoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
(2R)-2-amino-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
(3S,9aR)-3-benzyl-2-methyl-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 4-{[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}benzoate
3-({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
2-methyl-4-(5-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}thiophen-2-yl)but-3-yn-2-ol
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3-oxazolidin-2-one
2-amino-4-(1-benzofuran-2-yl)-6-(oxolane-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2S,4S)-4-amino-1-[4-(azepan-1-yl)-4-oxobutanoyl]-N-methylpyrrolidine-2-carboxamide
1-cyclopentanecarbonyl-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]piperidine-4-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
3-(azepane-1-carbonyl)-N,1-dimethyl-N-[2-(pyridin-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,5R)-3-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[2-(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-cyclohexyl-N-methyl-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyrrolidine-1-carbonyl)piperidine
1-(6-cyclopropylpyrimidin-4-yl)-4-(piperidine-1-sulfonyl)-1,4-diazepane
3-methyl-1-(2-methylpropyl)-4-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
N,N-diethyl-1-[(1s,4s)-4-[2-(2H-1,3-benzodioxol-5-yl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1,3,5-trimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrazole-4-carboxamide
3-(7-fluoro-2-methylquinoline-4-carbonyl)-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
5-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
N-[(3,4-dimethoxyphenyl)methyl]-2-(4-fluorophenyl)-N-(pyridin-2-ylmethyl)acetamide
1-(2-methoxy-6-methylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{2-[bis(2-hydroxyethyl)amino]ethyl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-ethyl-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-methyl-4-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)piperazin-2-one
2-chloro-4-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenol
3-[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[5-(2,3-dihydro-1-benzofuran-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{4-phenyl-1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-imidazol-5-yl}pyridine
(3S,4R)-1-(3-methoxybenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-(methoxymethyl)cyclobutane-1-carboxamide