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4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-6-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
(3R,4R)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-(2,3-dimethylphenyl)-N'-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]propanediamide
2-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-4,6-dimethylpyrimidine
5-({methyl[(3-{2-[4-(pyridine-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
2-{[methyl(quinolin-5-ylmethyl)amino]methyl}benzonitrile
3-methyl-5-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(propan-2-yl)amine
N,N-dimethyl-2-[(1S,5R)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-fluoro-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
1-[(1S,5R)-6-[(4-fluorophenyl)methanesulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-({4-[2-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
{4-[2-(3-methoxyphenoxy)ethyl]phenyl}methanamine
(1S,5R)-3-methyl-6-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
4-(2-amino-6-butanoyl-3-cyano-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl)benzoic acid
3-(2-oxo-2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethyl)-3,4-dihydroquinazolin-4-one
3-{5-[(2,3-difluoro-6-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-amino-3-ethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
7-(2-ethoxyacetyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-methyl-14-(6-phenoxypyridin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-(4-methanesulfonylphenyl)-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
4-(dimethyl-1,2-oxazol-4-yl)-3-(4-methyl-1H-imidazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-amino-2-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}ethan-1-ol
1-(2-chlorophenyl)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
1-cyclopentyl-N-methyl-5-oxo-N-[3-(1H-pyrazol-1-yl)propyl]pyrrolidine-3-carboxamide
2-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]thiolan-3-amine
(2R,3R)-3-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
N-[(3R,4R)-1-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(pyrrolidin-1-yl)pyrrolidine
2-ethyl-5-{1-[1-(4-methanesulfonylphenyl)ethyl]-1H-imidazol-2-yl}pyrimidine
N,6-dimethyl-N-[(2-methylpyridin-4-yl)methyl]-2-propylpyrimidin-4-amine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)propanamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,2-dimethylpropanamide
N-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}propanamide
(2R,3S,6R)-5-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}cyclopropanesulfonamide
methyl 2-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetate
2-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]-1H-1,2,3-triazol-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
N-butyl-N-methyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(morpholin-3-yl)ethan-1-one
1-(4-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-(1H-indol-5-ylmethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide