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3-(1-methyl-1H-pyrazol-5-yl)-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)propanamide
3-({[1-(naphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)propan-1-ol
1,3-dimethyl-N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]-1H-pyrazole-5-carboxamide
1-[2-(4-tert-butylphenoxymethyl)-4-hydroxypyrimidine-5-carbonyl]piperidine-3-carbonitrile
2-(4-methoxynaphthalen-1-yl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-(3-hydroxyazetidine-1-carbonyl)-6-(4-methoxyphenyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
3-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
methyl({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})(1,2-oxazol-3-ylmethyl)amine
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methyl-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
1-(2-fluoroethyl)-2-(8-methoxy-2H-chromen-3-yl)-1H-imidazole
2-[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amino]-N-(2,3-dimethylphenyl)acetamide
1-cyclopentyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{2-oxo-4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperazin-1-yl}benzonitrile
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyridin-3-ylmethyl)propanamide
7-[2-(ethylamino)pyrimidine-5-carbonyl]-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
5-methyl-N-(2-phenoxyethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-(2,3-dihydroxypropyl)-1-(2-methoxy-6-methylphenyl)-3-methylurea
6-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyridine-3-carboxamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
6-{[1-(4-fluorophenyl)ethyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(4-{2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethoxy}phenyl)propan-1-one
3-{[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
(3R,5S)-N3-(4-fluorophenyl)-N5-[(3-fluorophenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
2-(3-methoxypropyl)-8-[2-(1H-1,2,4-triazol-1-ylmethyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-[(3-methoxyphenyl)methyl]-8-(pyridazine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-cyclopropyl-1-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-4-methylpyrrolidin-2-one
4-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-5-ethyl-2-methylpyrimidine
N-[2-(4-chlorobenzenesulfonamido)ethyl]-3-cyclopropyl-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(7-methyl-1-benzofuran-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-amino-6-propyl-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2-(trifluoromethyl)morpholine
2-(5-{1-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)benzonitrile
N-(2,3-dihydro-1H-inden-2-yl)-4-(2-oxopyrrolidin-1-yl)-N-propylbenzamide
N-tert-butyl-2-[1-(cyclopropylmethyl)-1H-pyrazol-4-yl]benzene-1-sulfonamide
8-(2,2-dimethylpropyl)-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,8aR)-6-(1H-indazole-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-cyclopropyl-5-[(2,4-dimethoxy-3-methylphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
(1R,3S,5S)-8-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
(4aR,7aS)-N,N-dimethyl-4-(1-methyl-1H-pyrazole-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-(cyclopropylmethoxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(2-phenylethyl)-1,4-diazepan-2-one
1-(3-methoxypropyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-fluorophenyl)-3-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(3-ethoxyphenyl)methyl]amino}ethan-1-ol
2-(cyclopropylmethyl)-8-[(5-methoxy-1H-indazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3-{2-[1-(5-chloropyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
6-fluoro-N-methyl-N-[(6-methylpyridin-2-yl)methyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide