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2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
(1R,5S)-N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(2S,4S)-1-cyclopentyl-N,N-diethyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(prop-2-en-1-yl)piperidine-3-carboxamide
1-[(diethylcarbamoyl)methyl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[(3S,4R)-3-cyclopropyl-4-{[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}pyrrolidin-1-yl]acetamide
3,6-dimethyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(furan-2-yl)ethane-1,2-dione
1-(2-methoxyethyl)-3-methyl-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)pyridine-3-carboxylic acid
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
N-[3-(3-hydroxypiperidin-1-yl)propyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
ethyl(pyridin-3-ylmethyl)[2-(pyrrolidin-1-yl)ethyl]amine
5-[2-(4-methylpentyl)morpholine-4-carbonyl]-1H-1,2,3-benzotriazole
6-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinoxaline
(3aR,5R,6S,7aS)-2-[1-(pyrimidin-2-yl)piperidin-4-yl]-octahydro-1H-isoindole-5,6-diol
2-(2,5-dimethoxyphenyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
5-[({[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-amino-6-(pyridin-2-yl)-4-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
({2-[(2-chlorophenyl)methoxy]-7-fluoroquinolin-3-yl}methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
(3-{3-[3-(dimethyl-1,3-thiazol-5-yl)phenyl]-1H-pyrazol-1-yl}propyl)dimethylamine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
1-(morpholine-4-sulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-{[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}benzoic acid
7-(3-chlorophenyl)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-(2-methyl-1,3-thiazol-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(1H-pyrazol-1-ylmethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
N,N,4-trimethyl-3-{[(1-propylcyclopropyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
methyl 2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetate
3-(2-amino-1,3-thiazol-4-yl)-N-[(4-fluorophenyl)methyl]-N-(pyridin-2-ylmethyl)propanamide
1-cyano-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropane-1-carboxamide
4-[2-(4-chlorophenyl)morpholin-4-yl]quinoline
7-(3,4-dihydronaphthalen-2-yl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 2-{1-[3-(thiophen-3-yl)propanoyl]piperidin-2-yl}acetate
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
{1-[2-(4-chlorophenoxy)ethyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
1-{7-[(3-ethenylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methoxyethan-1-one
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-N-ethyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(3R,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
(2S)-2-amino-N-butyl-N-(furan-2-ylmethyl)-3-(1,3-thiazol-4-yl)propanamide
1-(1,4-dioxan-2-ylmethyl)-1-methyl-3-(2-phenylphenyl)urea
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
5-(2,6-dimethoxyphenyl)-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1,2,4-triazin-3-amine