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1-[2-(4-methoxyphenyl)ethyl]-4-[(pyridin-2-ylmethyl)amino]pyrrolidin-2-one
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-{5-[(1R,2R)-2-phenylcyclopropanecarbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
2-(4-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenoxy)ethan-1-ol
5-(2-chlorophenyl)-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]furan-2-carboxamide
3-(azepane-1-sulfonyl)-5-(2-cyanophenyl)benzoic acid
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxan-4-yl)pyridin-2-amine
2-{5-cyclopropyl-4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-methoxyphenyl)pyrimidine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2,3,4-trimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
(3R,5S)-5-(morpholine-4-carbonyl)-N-[2-(1,3-thiazol-4-yl)ethyl]piperidine-3-carboxamide
2-chloro-5-acetamido-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)benzamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole
N-methyl-2-[methyl(pyridin-4-ylmethyl)amino]-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
4-[4-(benzyloxy)-3-fluorophenyl]-7H-pyrrolo[2,3-d]pyrimidine
(4aS,8aR)-2-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-decahydroisoquinoline
N-(3-chloro-4-fluorophenyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carboxamide
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
2-(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)-3-methylpyrazine
N-[2-(dimethylamino)ethyl]-3-(2-hydroxyphenyl)-N-[(4-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
(1S,4S)-2-[3-(5-methylfuran-2-yl)benzoyl]-2,5-diazabicyclo[2.2.1]heptane
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
2-[(3-methoxyphenyl)amino]-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]butanamide
3-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)-N-(pyrazin-2-yl)benzamide
5-[(4,6-dimethylpyrimidin-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(5-methoxy-1H-indol-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
[2-(1H-imidazol-1-yl)ethyl](methyl)[2-methyl-2-(morpholin-4-yl)propyl]amine
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(3,4-dimethoxyphenyl)acetamide
7-fluoro-1-methyl-N-(1-methyl-1H-1,2,3-triazol-4-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
(1R,5R)-3-(pyridine-2-carbonyl)-6-[3-(1H-pyrrol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
1,9-dimethyl-4-(5-phenyl-1,3,4-thiadiazol-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-butyl-N-[(4-fluorophenyl)methyl]-4-methoxycyclohexane-1-carboxamide
(2S)-N2-ethyl-N1-[3-(pyridin-2-yl)phenyl]pyrrolidine-1,2-dicarboxamide
N-{[6-(5-chloro-2-methoxyphenyl)pyridin-3-yl]methyl}acetamide
4-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)pyrimidine
2-{[4-(1-phenylethyl)-5-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](4-methoxy-4-methylpentan-2-yl)amine
N-methyl-N-{2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]ethyl}methanesulfonamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(3-phenylphenyl)methyl]acetamide
1-{5-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
1-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-phenylpiperazine
3-[(3R,4S)-4-(dimethylamino)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-3-yl]propan-1-ol
1-[1-(1-benzofuran-2-ylmethyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methoxy]-1H-indole
N-cyclopropyl-1-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}piperidine-3-carboxamide