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7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1H-imidazol-2-ylmethyl)-2,7-diazaspiro[4.5]decane
3-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
5-(4-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
4-[1-(6-methoxypyrimidin-4-yl)piperidin-3-yl]-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
2-(2-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-cyclopropyl-1-{1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methylquinoxaline-5-carboxamide
(5-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}furan-2-yl)methanol
8-[2-(2-methoxy-4-methylphenoxy)ethyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(3-{[butyl(pyridin-3-ylmethyl)carbamoyl]amino}-4-fluorophenyl)propanamide
N-cyclopropyl-3-[(quinolin-2-ylmethyl)sulfamoyl]benzamide
N-(1-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
2-methyl-5-({2-[4-(pyridin-2-yl)phenyl]-1H-imidazol-1-yl}methyl)pyrazine
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(pyrrolidine-1-carbonyl)piperidine
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
1-[(4-fluorophenyl)methyl]-4-(3-fluoropyridin-4-yl)-1,4-diazepane
8-(2,6-dimethoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
6-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrazine-2-carboxamide
(2R)-2-{[2-(phenylamino)pyrimidin-5-yl]formamido}pentanediamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
(1S,5R)-6-(cyclobutylmethyl)-3-[(2-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylpyridine-3-carboxamide
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-(dimethylamino)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(3-methylphenyl)acetamide
1-(2-fluorophenyl)-2,2-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}cyclopropane-1-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[2-(3-fluorophenyl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-ethyl-1-methyl-3-{[1-(piperidine-1-sulfonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3,4-dimethylphenyl)-N-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2S)-4-methyl-2-(2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamido)pentanamide
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(pentan-3-yl)acetamide
1-(difluoromethyl)-N-(prop-2-en-1-yl)-N-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-ethyl-1-oxo-5-(pyridin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-ethyl-1-methyl-3-[1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(4-fluorophenyl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
3-[4-(2H-1,3-benzodioxol-5-yl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
3-(4-fluorophenyl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
6-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]pyrazine-2-carboxamide
2-{2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
6-{[4-(4-methyl-1,4-diazepane-1-carbonyl)piperidin-4-yl]oxy}quinoline
2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2-{2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-3-methylpyridin-4-amine
(3R,4R)-1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-({3-methyl-7-[2-(4-phenylphenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxane-4-carboxamide