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2-cyclopentyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
6-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2,2,6,6-tetramethyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]piperidin-4-amine
methyl (2S)-1-{2-[4-(4-{methyl[(3-methylpyridin-2-yl)methyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
2-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(1,3-thiazol-2-yl)ethyl]acetamide
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-(pyridin-2-yl)piperazine
N-[7-(3-benzoylpiperidine-1-carbonyl)-2-cyclobutyl-1-methyl-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
6-methyl-4-oxo-2-(2-phenylethyl)-N,N-bis(prop-2-en-1-yl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-chloro-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(2-methoxypyridin-3-yl)pyridin-3-yl]-2-methylpropanamide
N-({1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl}methyl)-2-(pyridin-4-yl)acetamide
N-{2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-2-yl}thiophene-2-carboxamide
5-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-methyl-1H-pyrazole
(1H-imidazol-2-ylmethyl)(methyl)(4-methyl-1-phenylpentyl)amine
1-(2-methoxy-4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
(2S)-1-{[(2-acetamidophenyl)carbamoyl]methyl}pyrrolidine-2-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-2-(methoxymethyl)-6-methyl-1-(3-phenylpropyl)-1,4-dihydropyridin-4-one
(1R,7S)-3-(2,2-dimethylpropyl)-6-(5-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(2S,4S)-4-amino-1-[2-(dimethyl-1,3-thiazol-4-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
N,5-dimethyl-N-(2-methylpropyl)-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl]propanoic acid
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazinan-2-yl)propanamide
2-[(1S,5R)-3-{[3-(2-aminoethyl)phenyl]methyl}-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(4-cyanopyridin-2-yl)piperidin-3-yl]propanamide
3-propyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dimethoxypyrimidine-4-carboxamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]urea
N-methyl-2-(pyrazin-2-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
4-(oxolane-2-carbonyl)-7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-methyl-1-(2-methylnaphthalen-1-yl)urea
1-(carbamoylmethyl)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
(3-{2-[1-(1H-indazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-[(2S)-oxolane-2-carbonyl]piperidine
3-({[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]amino}methyl)pyrrolidin-3-ol
2-(3,3-diphenylpiperidine-1-carbonyl)morpholine
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-[3-(trifluoromethyl)phenoxy]piperidine
N-cyclopropyl-1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3S)-1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]acetamide
5-cyclopropanecarbonyl-1'-(5-fluoropyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[4-(1-methoxyethyl)phenyl]-1-propyl-1H-1,2,4-triazole
1-{3-[2-(2,2-diphenylethyl)morpholin-4-yl]-3-oxopropyl}pyrrolidin-2-one
(1R,5R)-N,N-dimethyl-6-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinazolin-4-amine
1-(1-benzofuran-2-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
N-(2,2-difluoroethyl)-4-[(3-hydroxypiperidin-1-yl)sulfonyl]benzamide