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2-methyl-5-{[(3S,5R)-1-(pyridin-4-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methoxy}pyridine
(3R,7S,8aS)-3-(2-methylpropyl)-7-({[4-(propan-2-yl)phenyl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[9-acetyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-hydroxyethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(6-ethylpyrimidin-4-yl)pyrrolidin-3-yl]-4-methylpiperidine-4-carboxamide
2-{5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
3-(3-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methoxypyridazine
1-(3-methyl-1,2-oxazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methylbenzamide
5-ethyl-2-methyl-4-[3-(pyridin-4-yl)azetidin-1-yl]pyrimidine
{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
N-methyl-4-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(pyridin-3-yl)ethyl]benzamide
N-cyclohexyl-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-[(4aR,7aS)-4-[(4-ethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-[3-(1H-pyrazol-5-yl)phenyl]-1-(pyrimidin-5-ylmethyl)piperidine-4-carboxamide
2-methyl-5-(4-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
5-[(quinolin-8-yloxy)methyl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
3,7-dimethyl-8-[2-(trifluoromethyl)morpholin-4-yl]-2,3,6,7-tetrahydro-1H-purine-2,6-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-1H-indazole-3-carboxamide
8-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-6-oxo-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-(4,4-dimethyl-2-oxopyrrolidin-1-yl)-N-[2-(3-methoxyphenoxy)ethyl]-N-methylacetamide
3-(3-fluorophenyl)-N-methyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
4-methyl-3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}benzene-1-sulfonamide
{4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}methanol
2-[(3R,4R)-3-hydroxy-4-(morpholin-4-yl)piperidin-1-yl]pyridine-3-carboxamide
N-(1-methoxypropan-2-yl)-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidine-4-carboxamide
8-(1-methoxypropan-2-yl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(dimethylamino)-2-(3-methylphenyl)acetamide
3,3-dimethyl-1-(2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)urea
N-[1-(cyclohex-1-en-1-yl)ethyl]-7-methanesulfonyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2,4-dimethoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
2-{4-[1-(2-phenylethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}ethan-1-ol
6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
(2E)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-(furan-2-yl)-N-methylprop-2-enamide
5,6-dimethyl-3-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
2-ethyl-6-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrimidin-4-amine
1-[(4-fluorophenyl)methyl]-4-{[(5-methylthiophen-2-yl)methyl]amino}pyrrolidin-2-one
1-benzyl-3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-[4-(2,4-difluorophenyl)-1H-pyrazol-1-yl]-N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[4-(pyrimidin-5-yl)phenyl]methyl}piperidin-3-ol
N-(4-fluorophenyl)-3-{[(6-methylpyridin-3-yl)carbamoyl]methyl}morpholine-4-carboxamide
1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-4-(thiophen-3-ylmethyl)piperazine
4-{[5-(1-cyclopentanecarbonylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-methylquinoline-4-carboxamide
2-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(azepan-1-yl)-2-hydroxypropyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide