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1-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)cyclopropane-1-carboxamide
3-[(dimethylamino)methyl]-1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)piperidin-3-ol
(3R,5S)-N3-ethyl-N5-(4-methylphenyl)-N3-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
{1-[(1-ethyl-1H-indol-6-yl)methyl]pyrrolidin-3-yl}methanamine
1-(carbamoylmethyl)-N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]piperidine-3-carboxamide
N-cyclopropyl-1-[1-(5-methylpyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-(morpholin-4-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(pyridin-3-yl)acetamide
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(1-methylpiperidin-4-yl)methyl]piperazine
N-[2-(benzyloxy)ethyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1-ethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[2-(1H-imidazol-1-yl)acetamido]-N-(3-methoxyphenyl)benzamide
3-{[4-(3-hydroxyphenyl)piperazin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
ethyl 5-acetyl-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3R,7S,8aS)-7-({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}amino)-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
4-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
1-(4-fluorophenyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopropane-1-carboxamide
2-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
N-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(thian-4-yl)piperidin-4-amine
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
2-{9-[(2-chloro-4-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
2-[(3-methoxyphenyl)amino]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]butanamide
N-{[(2S,4S)-4-fluoro-1-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)pyrrolidin-2-yl]methyl}methanesulfonamide
1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}azepan-2-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
ethyl 1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidine-2-carboxylate
N-{1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
1-(2,3-dihydro-1H-inden-5-yl)-3-(oxolan-3-yl)-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazole
6-fluoro-4-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-[1-(2-methylpropyl)-1H-pyrazol-5-yl]acetamide
6-methyl-2-(3-methyl-1H-pyrazole-4-carbonyl)-5-[5-(1-methylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-3-amine
3-{5-[(4-methyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(2-phenylethyl)acetamide
(3R,4R)-1-(3-methylfuran-2-carbonyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-2-one
1-(4,6-dimethylpyrimidin-2-yl)-N-[3-(1H-imidazol-2-yl)propyl]piperidin-4-amine
N-cyclopentyl-5-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{2-methyl-6-[1-(2-propoxyethyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
3-(1H-imidazol-2-yl)-N-[(1R,2S)-2-phenylcyclopropyl]benzamide
6-(methoxymethyl)-N-{1-oxaspiro[4.4]nonan-3-yl}pyrimidin-4-amine
2-(5-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}furan-2-yl)benzonitrile
3-(hydroxymethyl)-N-(3-methylcinnolin-5-yl)piperidine-1-carboxamide
2-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]benzamide
1-methyl-4-(2-{[6-(2-methyl-1H-imidazol-1-yl)pyridazin-3-yl]oxy}hex-5-en-1-yl)-1,4-diazepane
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-(2-methoxyphenyl)acetamide