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2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methylacetamide
7-[(3,4-difluorophenyl)methyl]-2-(3-methoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N5-butyl-N3-cyclohexyl-1-(furan-2-ylmethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-(4-methylpiperazine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(adamantan-2-yl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
4-ethyl-1-(oxolan-2-ylmethyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(cyclopropylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
3-[(4,4-diphenylpiperidin-1-yl)methyl]-3-hydroxy-1-methylpiperidin-2-one
1-[4-(4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
[(2S)-1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
9-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
7-(4-aminopyrimidin-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(2-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5-(1H-indol-1-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
5-({[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-1-methyl-1H-1,2,3,4-tetrazole
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methylfuran-2-carboxamide
1-cyclopropyl-N-[(4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-methylphenol
4-(5-acetylthiophene-3-carbonyl)-3-benzylpiperazin-2-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-{4-[1-(N-methyl-1-thiophen-3-ylformamido)-2-phenylethyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
N-{[1-cyclohexyl-3-(3,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}methanesulfonamide
1-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]butane-1,2-dione
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
N-benzyl-1-[1-(pent-4-enoyl)piperidin-4-yl]piperidine-3-carboxamide
2-{3-[3-(6-methylpyridin-3-yl)phenyl]-1H-pyrazol-1-yl}-N-(oxolan-2-ylmethyl)acetamide
N-benzyl-N-(2-hydroxyethyl)-5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-(prop-2-en-1-yl)-4-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]pyrrolidin-2-one
2-methyl-N-[2-(pyridin-3-yl)ethyl]-1-benzofuran-5-carboxamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
5-{[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
N-{2-[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridin-3-amine
4-[(4-fluorophenyl)methyl]-1-(2-methylpyrimidine-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-hydroxy-3-(2-methylphenoxy)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
1'-(1-methyl-1H-pyrazole-3-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-methyl-1-({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)-1,4-diazepan-5-one
(1R,5S,6S)-6-({4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
{1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-3-propylpiperidin-3-yl}methanol
1'-(1-benzofuran-2-ylmethyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]-2-(2-methylphenyl)acetic acid
3-{1-[4-(1-hydroxyethyl)phenyl]-3,5-dimethyl-1H-pyrazol-4-yl}propanoic acid
(1S,5R)-6-benzyl-3-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(4-fluorophenyl)-4-oxobutanamido]acetic acid
2-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-N,N-dimethylaniline
3-{1-[(6-ethoxypyridin-3-yl)methyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-tert-butyl-6-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
5-ethyl-1'-(5-methyl-1H-indole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]