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(2S)-N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}pyrrolidine-2-carboxamide
N-({8-[2-(3,4,5-trimethoxyphenyl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-2-carboxamide
N-[(1,4-dimethylpiperazin-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-methoxy-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)acetamide
N-cyclopropyl-1-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
7-(3-chlorophenyl)-4-(6-cyclopropylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-chloropyridine-4-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
4-(5-oxo-1-propylpyrrolidin-3-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(1-benzofuran-3-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
4-(7-chloroquinolin-4-yl)-2-({[2-(diethylamino)ethyl](methyl)amino}methyl)phenol
(3S,4S)-4-(morpholin-4-yl)-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}thiolan-3-amine
(5-{[4-(dimethylamino)phenyl]methyl}-1-methyl-1H-1,2,4-triazol-3-yl)(phenyl)methanol
(3R,4R)-1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
4-[1-(1,4-dioxan-2-ylmethyl)-1H-imidazol-2-yl]-2-methoxy-6-(prop-2-en-1-yl)phenol
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2-methoxyethyl)-2-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-(oxolan-2-ylmethyl)-9-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-2-phenyl-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-(1-{[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-cyclopentyl-5-(1-methyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3,4-dimethoxypyridin-2-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
ethyl 4-{[4-(3-methoxyphenyl)phenyl]carbamoyl}piperazine-1-carboxylate
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[4-(cyclohex-3-en-1-ylmethyl)piperazin-1-yl]-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-methyl-2-(4-methyl-1H-imidazol-5-yl)-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
N-{[1-(dimethylamino)cyclohexyl]methyl}-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
3-(3-aminopyrrolidine-1-carbonyl)-N-[(2-methylpyridin-4-yl)methyl]benzene-1-sulfonamide
4-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-1,2-dimethylpiperazine
2-[4-(2-aminopyrimidin-4-yl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[(2-fluorophenyl)methyl]-3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
3-methyl-N-{1-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
2-ethoxy-6-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]phenol
dimethyl({[4-methyl-5-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,4-dimethyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
4-{4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]phenyl}-2-methylbutan-2-ol
2-(1-methyl-1H-pyrrole-2-carbonyl)-8-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
3-{2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}propanamide
(3S,4S)-1-[(6-chloroquinolin-2-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
(3R,4S)-4-{[(3-chloro-4,5-diethoxyphenyl)methyl](ethyl)amino}oxolan-3-ol
(3S)-1-{1-methyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[2-(piperidin-1-yl)ethyl]propanamide
3-(1H-imidazol-1-ylmethyl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-[4-(cyclopropylmethoxy)phenyl]-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide