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ethyl 2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]pyridine-3-carboxylate
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
1-methyl-N-[4-(pyridin-2-yl)butyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,9aR)-N-[2-(4-sulfamoylphenyl)ethyl]-octahydro-1H-quinolizine-1-carboxamide
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
(3R,5S)-1-benzyl-N-(3-methoxypropyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
[2-(2-amino-9H-purin-6-yl)phenyl]methanol
1,3-dimethyl-6-(pyridin-2-yl)-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-(3-chloro-4-methylbenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[1-(3-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-3-methoxypropanamide
(3aR,6aR)-2-(oxane-4-carbonyl)-5-(pyridin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,4S)-1-acetyl-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
N'1-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]cyclopropane-1,1-dicarboxamide
N,N-dimethyl-2-[(1S,5R)-6-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
[(3R,4R)-1-(5-chloro-2-methylpyrimidine-4-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-[5-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
5-methoxy-2-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-4-ol
1-(2-aminoethyl)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{1-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-(azepan-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
N-(1-{1-[(2S)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N'-(3,5-dimethylphenyl)-N-methyl-N-[3-(oxolan-2-yl)propyl]propanediamide
3-propoxy-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine
1-({5-[(4-tert-butylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N,2-dimethyl-N-(1-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-2-phenylethyl)furan-3-carboxamide
5-fluoro-2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyridine
1-{1-[(2-ethoxynaphthalen-1-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
4-[1-(2-methoxyacetyl)piperidine-4-carbonyl]-3-methyl-1-phenylpiperazin-2-one
(2S,4S)-4-cyclopentaneamido-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methylpyrrolidine-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-[4-(methylsulfanyl)phenyl]acetamide
2-(2-fluoro-5-methylphenyl)pyridine-4-carboxamide
methyl 4-methyl-2-{2-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]acetamido}-1,3-thiazole-5-carboxylate
(3aR,6aR)-2-[2-(2,4-dimethylphenoxy)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-3-(2-methoxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
6-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]-N,1-dimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(2S,4R)-4-{[(4-chlorophenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
(2R)-2-amino-1-(4-ethyl-3,3-dimethylpiperazin-1-yl)-3-(ethylsulfanyl)propan-1-one
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazole
7-methyl-2-(2-{[(2-methylphenyl)methyl]sulfanyl}acetyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4S)-1-cyclobutanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
1'-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(methylsulfanyl)ethan-1-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}pyridine-3-carboxamide
8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione